日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Use of Informer Sets in Screening: Perspectives on an Efficient Strategy to Identify New Probes

筛选中使用信息集:识别新探针的有效策略观点

Paul A Clemons, Joshua A Bittker, Florence F Wagner, Allison Hands, Vlado Dančík, Stuart L Schreiber, Amit Choudhary, Bridget K Wagner

Postnatal Acetaminophen and Potential Risk of Autism Spectrum Disorder among Males

产后服用对乙酰氨基酚与男性患自闭症谱系障碍的潜在风险

Bittker, Seth S; Bell, Kathleen R

The Carcinogenome Project: In Vitro Gene Expression Profiling of Chemical Perturbations to Predict Long-Term Carcinogenicity

致癌基因组计划:通过化学扰动的体外基因表达谱预测长期致癌性

Amy Li, Xiaodong Lu, Ted Natoli, Joshua Bittker, Nisha S Sipes, Aravind Subramanian, Scott Auerbach, David H Sherr, Stefano Monti

GDC-0879, a BRAFV600E Inhibitor, Protects Kidney Podocytes from Death

GDC-0879,一种 BRAFV600E 抑制剂,可保护肾足细胞免于死亡

Jonas Sieber, Nicolas Wieder, Abbe Clark, Manuel Reitberger, Sofia Matan, Jeannine Schoenfelder, Jianming Zhang, Anna Mandinova, Joshua Adam Bittker, Juan Gutierrez, Ozan Aygün, Namrata Udeshi, Steven Carr, Peter Mundel, Andreas Werner Jehle, Anna Greka

High Throughput Screen Identifies Interferon γ-Dependent Inhibitors of Toxoplasma gondii Growth

高通量筛选鉴定出干扰素γ依赖性的弓形虫生长抑制剂

Joshua B Radke, Kimberly L Carey, Subrata Shaw, Shailesh R Metkar, Carol Mulrooney, Jennifer P Gale, Joshua A Bittker, Robert Hilgraf, Eamon Comer, Stuart L Schreiber, Herbert W Virgin, Jose R Perez, L David Sibley

High-Throughput Screens To Identify Autophagy Inducers That Function by Disrupting Beclin 1/Bcl-2 Binding

通过高通量筛选鉴定通过破坏 Beclin 1/Bcl-2 结合发挥作用的自噬诱导剂

Wei-Chung Chiang, Yongjie Wei, Yi-Chun Kuo, Shuguang Wei, Anwu Zhou, Zhongju Zou, Jenna Yehl, Matthew J Ranaghan, Adam Skepner, Joshua A Bittker, Jose R Perez, Bruce A Posner, Beth Levine

The Drug Repurposing Hub: a next-generation drug library and information resource

药物再利用中心:下一代药物图书馆和信息资源

Steven M Corsello, Joshua A Bittker, Zihan Liu, Joshua Gould, Patrick McCarren, Jodi E Hirschman, Stephen E Johnston, Anita Vrcic, Bang Wong, Mariya Khan, Jacob Asiedu, Rajiv Narayan, Christopher C Mader, Aravind Subramanian, Todd R Golub

Selective Chemical Inhibition of PGC-1α Gluconeogenic Activity Ameliorates Type 2 Diabetes

选择性化学抑制 PGC-1α 糖异生活性可改善 2 型糖尿病

Kfir Sharabi, Hua Lin, Clint D J Tavares, John E Dominy, Joao Paulo Camporez, Rachel J Perry, Roger Schilling, Amy K Rines, Jaemin Lee, Marc Hickey, Melissa Bennion, Michelle Palmer, Partha P Nag, Joshua A Bittker, José Perez, Mark P Jedrychowski, Umut Ozcan, Steve P Gygi, Theodore M Kamenecka, Gera

A dataset of images and morphological profiles of 30 000 small-molecule treatments using the Cell Painting assay

利用细胞染色分析法,构建了一个包含30000个小分子处理样本的图像和形态学特征的数据集。

Bray, Mark-Anthony; Gustafsdottir, Sigrun M; Rohban, Mohammad H; Singh, Shantanu; Ljosa, Vebjorn; Sokolnicki, Katherine L; Bittker, Joshua A; Bodycombe, Nicole E; Dancík, Vlado; Hasaka, Thomas P; Hon, Cindy S; Kemp, Melissa M; Li, Kejie; Walpita, Deepika; Wawer, Mathias J; Golub, Todd R; Schreiber, Stuart L; Clemons, Paul A; Shamji, Alykhan F; Carpenter, Anne E

Small-molecule inhibitors directly target CARD9 and mimic its protective variant in inflammatory bowel disease

小分子抑制剂直接靶向 CARD9 并模仿其在炎症性肠病中的保护性变体

Elizaveta S Leshchiner, Jason S Rush, Michael A Durney, Zhifang Cao, Vlado Dančík, Benjamin Chittick, Huixian Wu, Adam Petrone, Joshua A Bittker, Andrew Phillips, Jose R Perez, Alykhan F Shamji, Virendar K Kaushik, Mark J Daly, Daniel B Graham, Stuart L Schreiber, Ramnik J Xavier