日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A dataset of images and morphological profiles of 30 000 small-molecule treatments using the Cell Painting assay

利用细胞染色分析法,构建了一个包含30000个小分子处理样本的图像和形态学特征的数据集。

Bray, Mark-Anthony; Gustafsdottir, Sigrun M; Rohban, Mohammad H; Singh, Shantanu; Ljosa, Vebjorn; Sokolnicki, Katherine L; Bittker, Joshua A; Bodycombe, Nicole E; Dancík, Vlado; Hasaka, Thomas P; Hon, Cindy S; Kemp, Melissa M; Li, Kejie; Walpita, Deepika; Wawer, Mathias J; Golub, Todd R; Schreiber, Stuart L; Clemons, Paul A; Shamji, Alykhan F; Carpenter, Anne E

Diversity-oriented synthesis yields novel multistage antimalarial inhibitors.

多样性导向合成产生新型多阶段抗疟疾抑制剂

Kato Nobutaka, Comer Eamon, Sakata-Kato Tomoyo, Sharma Arvind, Sharma Manmohan, Maetani Micah, Bastien Jessica, Brancucci Nicolas M, Bittker Joshua A, Corey Victoria, Clarke David, Derbyshire Emily R, Dornan Gillian L, Duffy Sandra, Eckley Sean, Itoe Maurice A, Koolen Karin M J, Lewis Timothy A, Lui Ping S, Lukens Amanda K, Lund Emily, March Sandra, Meibalan Elamaran, Meier Bennett C, McPhail Jacob A, Mitasev Branko, Moss Eli L, Sayes Morgane, Van Gessel Yvonne, Wawer Mathias J, Yoshinaga Takashi, Zeeman Anne-Marie, Avery Vicky M, Bhatia Sangeeta N, Burke John E, Catteruccia Flaminia, Clardy Jon C, Clemons Paul A, Dechering Koen J, Duvall Jeremy R, Foley Michael A, Gusovsky Fabian, Kocken Clemens H M, Marti Matthias, Morningstar Marshall L, Munoz Benito, Neafsey Daniel E, Sharma Amit, Winzeler Elizabeth A, Wirth Dyann F, Scherer Christina A, Schreiber Stuart L

Advancing Biological Understanding and Therapeutics Discovery with Small-Molecule Probes

利用小分子探针推进生物学理解和治疗药物发现

Schreiber, Stuart L; Kotz, Joanne D; Li, Min; Aubé, Jeffrey; Austin, Christopher P; Reed, John C; Rosen, Hugh; White, E Lucile; Sklar, Larry A; Lindsley, Craig W; Alexander, Benjamin R; Bittker, Joshua A; Clemons, Paul A; de Souza, Andrea; Foley, Michael A; Palmer, Michelle; Shamji, Alykhan F; Wawer, Mathias J; McManus, Owen; Wu, Meng; Zou, Beiyan; Yu, Haibo; Golden, Jennifer E; Schoenen, Frank J; Simeonov, Anton; Jadhav, Ajit; Jackson, Michael R; Pinkerton, Anthony B; Chung, Thomas D Y; Griffin, Patrick R; Cravatt, Benjamin F; Hodder, Peter S; Roush, William R; Roberts, Edward; Chung, Dong-Hoon; Jonsson, Colleen B; Noah, James W; Severson, William E; Ananthan, Subramaniam; Edwards, Bruce; Oprea, Tudor I; Conn, P Jeffrey; Hopkins, Corey R; Wood, Michael R; Stauffer, Shaun R; Emmitte, Kyle A

Evolving BioAssay Ontology (BAO): modularization, integration and applications

生物测定本体(BAO)的演进:模块化、集成和应用

Abeyruwan, Saminda; Vempati, Uma D; Küçük-McGinty, Hande; Visser, Ubbo; Koleti, Amar; Mir, Ahsan; Sakurai, Kunie; Chung, Caty; Bittker, Joshua A; Clemons, Paul A; Brudz, Steve; Siripala, Anosha; Morales, Arturo J; Romacker, Martin; Twomey, David; Bureeva, Svetlana; Lemmon, Vance; Schürer, Stephan C

An Overview of the Challenges in Designing, Integrating, and Delivering BARD: A Public Chemical-Biology Resource and Query Portal for Multiple Organizations, Locations, and Disciplines

BARD(面向多个组织、地点和学科的公共化学生物学资源和查询门户)的设计、集成和交付所面临的挑战概述

de Souza, Andrea; Bittker, Joshua A; Lahr, David L; Brudz, Steve; Chatwin, Simon; Oprea, Tudor I; Waller, Anna; Yang, Jeremy J; Southall, Noel; Guha, Rajarshi; Schürer, Stephan C; Vempati, Uma D; Southern, Mark R; Dawson, Eric S; Clemons, Paul A; Chung, Thomas D Y

An interactive resource to identify cancer genetic and lineage dependencies targeted by small molecules

一个用于识别小分子靶向的癌症遗传和谱系依赖性的交互式资源

Basu, Amrita; Bodycombe, Nicole E; Cheah, Jaime H; Price, Edmund V; Liu, Ke; Schaefer, Giannina I; Ebright, Richard Y; Stewart, Michelle L; Ito, Daisuke; Wang, Stephanie; Bracha, Abigail L; Liefeld, Ted; Wawer, Mathias; Gilbert, Joshua C; Wilson, Andrew J; Stransky, Nicolas; Kryukov, Gregory V; Dancik, Vlado; Barretina, Jordi; Garraway, Levi A; Hon, C Suk-Yee; Munoz, Benito; Bittker, Joshua A; Stockwell, Brent R; Khabele, Dineo; Stern, Andrew M; Clemons, Paul A; Shamji, Alykhan F; Schreiber, Stuart L

Overcoming fluconazole resistance in Candida albicans clinical isolates with tetracyclic indoles

利用四环吲哚克服白色念珠菌临床分离株对氟康唑的耐药性

Youngsaye, Willmen; Dockendorff, Chris; Vincent, Benjamin; Hartland, Cathy L; Bittker, Joshua A; Dandapani, Sivaraman; Palmer, Michelle; Whitesell, Luke; Lindquist, Susan; Schreiber, Stuart L; Munoz, Benito

Piperazinyl quinolines as chemosensitizers to increase fluconazole susceptibility of Candida albicans clinical isolates

哌嗪基喹啉类化合物作为化学增敏剂可提高白色念珠菌临床分离株对氟康唑的敏感性

Youngsaye, Willmen; Vincent, Benjamin; Hartland, Cathy L; Morgan, Barbara J; Buhrlage, Sara J; Johnston, Stephen; Bittker, Joshua A; MacPherson, Lawrence; Dandapani, Sivaraman; Palmer, Michelle; Whitesell, Luke; Lindquist, Susan; Schreiber, Stuart L; Munoz, Benito

Directed evolution of protein enzymes using nonhomologous random recombination

利用非同源随机重组进行蛋白质酶的定向进化

Bittker, Joshua A; Le, Brian V; Liu, Jane M; Liu, David R

Nucleic acid evolution and minimization by nonhomologous random recombination

非同源随机重组介导的核酸进化与最小化

Bittker, Joshua A; Le, Brian V; Liu, David R