The Identification and Pharmacological Characterization of 6-(tert-Butylsulfonyl)-N-(5-fluoro-1H-indazol-3-yl)quinolin-4-amine (GSK583), a Highly Potent and Selective Inhibitor of RIP2 Kinase
6-(叔丁基磺酰基)-N-(5-氟-1H-吲唑-3-基)喹啉-4-胺 (GSK583) 的鉴定和药理学特性,一种高效且选择性的 RIP2 激酶抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.6b00211
Pamela A Haile, Bartholomew J Votta, Robert W Marquis, Michael J Bury, John F Mehlmann, Robert Singhaus Jr, Adam K Charnley, Ami S Lakdawala, Máire A Convery, David B Lipshutz, Biva M Desai, Barbara Swift, Carol A Capriotti, Scott B Berger, Mukesh K Mahajan, Michael A Reilly, Elizabeth J Rivera, Hel