A new strategy for hit generation: Novel in cellulo active inhibitors of CYP121A1 from Mycobacterium tuberculosis via a combined X-ray crystallographic and phenotypic screening approach (XP screen)
生成有效化合物的新策略:通过结合 X 射线晶体学和表型筛选方法(XP 筛选)寻找结核分枝杆菌 CYP121A1 的新型纤维素活性抑制剂
期刊:European Journal of Medicinal Chemistry
影响因子:6
doi:10.1016/j.ejmech.2022.114105
Martyn Frederickson, Irwin R Selvam, Dimitrios Evangelopoulos, Kirsty J McLean, Mona M Katariya, Richard B Tunnicliffe, Bethany Campbell, Madeline E Kavanagh, Sitthivut Charoensutthivarakul, Richard T Blankley, Colin W Levy, Luiz Pedro S de Carvalho, David Leys, Andrew W Munro, Anthony G Coyne, Chri