Selective inhibitors of SARM1 targeting an allosteric cysteine in the autoregulatory ARM domain
针对自调节 ARM 结构域中的变构半胱氨酸的 SARM1 选择性抑制剂
期刊:Proceedings of the National Academy of Sciences of the United States of America
影响因子:
doi:10.1073/pnas.2208457119
Hannah C Feldman, Elisa Merlini, Carlos Guijas, Kristen E DeMeester, Evert Njomen, Ellen M Kozina, Minoru Yokoyama, Ekaterina Vinogradova, Holly T Reardon, Bruno Melillo, Stuart L Schreiber, Andrea Loreto, Jacqueline L Blankman, Benjamin F Cravatt