日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Oseltamivir aziridines are potent influenza neuraminidase inhibitors and imaging agents

奥司他韦氮丙啶类药物是强效的流感神经氨酸酶抑制剂和显像剂。

Vriends, Merijn B L; Moran, Elisha; Calvelo, Martín; Hansen, Thomas; Pickles, Isabelle B; Xin, Xincheng; Biezeno, Marieke; Armstrong, Zachary W B; Ferraz, Maria J; Li, Lei; Lilley, Alice; Harvey, Ruth; Filippov, Dmitri V; Liao, Qinghua; Schröder, Sybrin P; van der Marel, Gijsbert A; Artola, Marta; Aerts, Johannes M F G; Blaza, James N; Codée, Jeroen D C; Rovira, Carme; Overkleeft, Herman S; Davies, Gideon J

Insights from aquaporin structures into drug-resistant sleeping sickness

从水通道蛋白结构中揭示耐药性昏睡病的机制

Matusevicius, Modestas; Corey, Robin A; Gragera, Marcos; Yamashita, Keitaro; Sprenger, Teresa; Ungogo, Marzuq; Blaza, James N; Castro-Hartmann, Pablo; Chirgadze, Dimitri Y; Chaitanya Vedithi, Sundeep; Afanasyev, Pavel; Melero, Roberto; Warshamanage, Rangana; Gusach, Anastasiia; Carazo, José-Maria; Carrington, Mark; Blundell, Tom; Murshudov, Garib N; Stansfeld, Phillip J; Sansom, Mark S P; De Koning, Harry P; Tate, Christopher G; Weyand, Simone

Remission spectroscopy resolves the mechanism of action of bedaquiline within living mycobacteria

反射光谱法解析了贝达喹啉在活分枝杆菌中的作用机制

Harrison, Suzanna H; Walters, Rowan C; Cheung, Chen-Yi; Springett, Roger J; Cook, Gregory M; Osman, Morwan M; Blaza, James N

Early activation of bioenergetic metabolism powers bacterial spore germination

生物能量代谢的早期激活为细菌孢子萌发提供动力

Gupta, Pooja; Caldbeck, Rebecca; Walters, Rowan C; Wells, Elodie C; Hardman, Bethany L; Christie, Graham; Springett, Roger J; Blaza, James N

Penton blooming, a conserved mechanism of genome delivery used by disparate microviruses.

Penton 膜破裂,是不同微病毒所采用的一种保守的基因组传递机制

Bardy Pavol, MacDonald Conor I W, Kirchberger Paul C, Jenkins Huw T, Botka Tibor, Byrom Lewis, Alim Nawshin T B, Traore Daouda A K, Koenig Hannah C, Nicholas Tristan R, Chechik Maria, Hart Samuel J, Turkenburg Johan P, Blaza James N, Beatty J Thomas, Fogg Paul C M, Antson Alfred A

Structural unification of diverse transmembrane acyltransferases reveals a conserved fold for the transmembrane acyl transferase (TmAT) superfamily

多种跨膜酰基转移酶的结构统一性揭示了跨膜酰基转移酶(TmAT)超家族的保守折叠结构。

Kinniment-Williams, Bethan E; Jurgeleviciute, Vytaute; West, Daniel T; Herman, Reyme; Blaza, James N; van der Woude, Marjan W; Thomas, Gavin H

A new family of bacterial ribosome hibernation factors

一个新的细菌核糖体冬眠因子家族

Karla Helena-Bueno #, Mariia Yu Rybak #, Chinenye L Ekemezie, Rudi Sullivan, Charlotte R Brown, Charlotte Dingwall, Arnaud Baslé, Claudia Schneider, James P R Connolly, James N Blaza, Bálint Csörgő, Patrick J Moynihan, Matthieu G Gagnon, Chris H Hill, Sergey V Melnikov

Mitochondrial DNA mutations drive aerobic glycolysis to enhance checkpoint blockade response in melanoma

线粒体DNA突变驱动有氧糖酵解,从而增强黑色素瘤中的检查点阻断反应

Mahnoor Mahmood,Eric Minwei Liu,Amy L Shergold,Elisabetta Tolla,Jacqueline Tait-Mulder,Alejandro Huerta-Uribe,Engy Shokry,Alex L Young,Sergio Lilla,Minsoo Kim,Tricia Park,Sonia Boscenco,Javier L Manchon,Crístina Rodríguez-Antona,Rowan C Walters,Roger J Springett,James N Blaza,Louise Mitchell,Karen Blyth,Sara Zanivan,David Sumpton,Edward W Roberts,Ed Reznik,Payam A Gammage  0

Cryo-EM structure of the CDK2-cyclin A-CDC25A complex

CDK2-细胞周期蛋白 A-CDC25A 复合物的低温电子显微镜结构

Rhianna J Rowland, Svitlana Korolchuk, Marco Salamina, Natalie J Tatum, James R Ault, Sam Hart, Johan P Turkenburg, James N Blaza, Martin E M Noble, Jane A Endicott

A promiscuous mechanism to phase separate eukaryotic carbon fixation in the green lineage.

绿色植物谱系中真核生物碳固定的相分离机制

Barrett James, Naduthodi Mihris I S, Mao Yuwei, Dégut Clément, Musiał Sabina, Salter Aidan, Leake Mark C, Plevin Michael J, McCormick Alistair J, Blaza James N, Mackinder Luke C M