Exploiting the 2-(1,3,4,9-tetrahydropyrano[3,4-b]indol-1-yl)acetic Acid Scaffold to Generate COXTRANs: A New Class of Dual Cyclooxygenase Inhibitors-Thromboxane Receptor Antagonists
利用 2-(1,3,4,9-四氢吡喃并[3,4-b]吲哚-1-基)乙酸骨架生成 COXTRANs:一类新型双重环氧合酶抑制剂-血栓素受体拮抗剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c02068
Blua, Federica; Boccato, Francesca; Buccellati, Carola; Risè, Patrizia; Barbieri, Silvia; Castiglioni, Laura; Balzulat, Annika; Rolando, Barbara; Marini, Elisabetta; Balestra, Marta; Introvigne, Maria Luisa; Giorgis, Marta; Sironi, Luigi; Tacconelli, Stefania; Hiesinger, Kerstin; Patrignani, Paola; Schmidtko, Achim; Steinhilber, Dieter; Proschak, Ewgenij; Sala, Angelo; Rovati, G Enrico; Bertinaria, Massimo