日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Novel Class of Complement 3a Receptor Agonists and Antagonists Derived from the TLQP-21 Peptide

一类源自TLQP-21肽的新型补体3a受体激动剂和拮抗剂

Rodriguez, Pedro; Pallais, Jean Pierre; He, Rongjun; Razzoli, Maria; McKee, John L; Bock, Hailey A; McCorvy, John D; Sham, Yuk Y; DiMarchi, Richard; Bartolomucci, Alessandro

Potent and Selective Human 5-HT(2B) Serotonin Receptor Antagonists: 4'-Cyano-(N)-methanocarba-adenosines by Synthetic Serendipity

合成意外发现的高效选择性人5-HT(2B)血清素受体拮抗剂:4'-氰基-(N)-甲氧基碳酰胺腺苷

Tosh, Dilip K; Pavan, Matteo; Clark, Allison A; Lammers, Josie; Villano, Serafina; Marri, Silvia; Sgambellone, Silvia; Choi, Suebin; Lee, Jihyun; Ivancich, Marko S; Bock, Hailey A; Campbell, Ryan G; Lewicki, Sarah A; Levitan, Ian M; Chen, Eric; Liu, Naili; Demby, Tamar; Gavrilova, Oksana; Gao, Zhan-Guo; Lucarini, Laura; McCorvy, John D; Jacobson, Kenneth A

Bioisosteric analogs of MDMA: Improving the pharmacological profile?

MDMA的生物等排体类似物:能否改善其药理特性?

Alberto-Silva Ana Sofia, Hemmer Selina, Bock Hailey A, da Silva Leticia Alves, Scott Kenneth R, Kastner Nina, Bhatt Manan, Niello Marco, Jäntsch Kathrin, Kudlacek Oliver, Bossi Elena, Stockner Thomas, Meyer Markus R, McCorvy John D, Brandt Simon D, Kavanagh Pierce, Sitte Harald H

N-(4-Bromo-2,5-Dimethoxyphenethyl)-6-(4-Phenylbutoxy)Hexan-1-Amine (XOB): A Novel Phenylalkylamine Antagonist of Serotonin 2A Receptors and Voltage-Gated Sodium Channels.

N-(4-溴-2,5-二甲氧基苯乙基)-6-(4-苯基丁氧基)己烷-1-胺 (XOB):一种新型的血清素 2A 受体和电压门控钠通道的苯烷基胺拮抗剂

Denomme Nicholas, Hernandez Ciria C, Bock Hailey A, Ohana Rachel F, Bakshi Shreeya, Sherwood Alexander M, McCorvy John D, Daley Paul F, Callaway Wyeth B, Hull Jacob M, Alt Andrew, Isom Lori L, Cozzi Nicholas V

Bioisosteric analogs of MDMA with improved pharmacological profile

具有改进药理特性的MDMA生物等排体类似物

Alberto-Silva, Ana Sofia; Hemmer, Selina; Bock, Hailey A; Alves da Silva, Leticia; Scott, Kenneth R; Kastner, Nina; Bhatt, Manan; Niello, Marco; Jäntsch, Kathrin; Kudlacek, Oliver; Bossi, Elena; Stockner, Thomas; Meyer, Markus R; McCorvy, John D; Brandt, Simon D; Kavanagh, Pierce; Sitte, Harald H

Pharmacological Mechanism of the Non-hallucinogenic 5-HT(2A) Agonist Ariadne and Analogs

非致幻性 5-HT(2A) 激动剂 Ariadne 及其类似物的药理机制

Cunningham, Michael J; Bock, Hailey A; Serrano, Inis C; Bechand, Benjamin; Vidyadhara, D J; Bonniwell, Emma M; Lankri, David; Duggan, Priscilla; Nazarova, Antonina L; Cao, Andrew B; Calkins, Maggie M; Khirsariya, Prashant; Hwu, Christopher; Katritch, Vsevolod; Chandra, Sreeganga S; McCorvy, John D; Sames, Dalibor