日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Evaluation of the Functional Suitability of Carboxylate Chlorin e(6) Derivatives for Use in Radionuclide Diagnostics

羧酸氯e(6)衍生物在放射性核素诊断中的功能适用性评价

Larkina, Mariia; Demina, Anastasia; Suvorov, Nikita; Ostroverkhov, Petr; Plotnikov, Evgenii; Varvashenya, Ruslan; Bodenko, Vitalina; Yanovich, Gleb; Prach, Anastasia; Pogorilyy, Viktor; Tikhonov, Sergey; Popov, Alexander; Usachev, Maxim; Volel, Beatrice; Vasil'ev, Yuriy; Belousov, Mikhail; Grin, Mikhail

Evaluation of a novel (177)Lu-labelled therapeutic Affibody molecule with a deimmunized ABD domain and improved biodistribution profile

对一种新型的(177)Lu标记的治疗性Affibody分子进行评估,该分子具有去免疫化的ABD结构域和改进的生物分布特征。

Liu, Yongsheng; Oroujeni, Maryam; Liao, Yunqi; Vorobyeva, Anzhelika; Bodenko, Vitalina; Orlova, Anna; Konijnenberg, Mark; Carlqvist, Matilda; Wahlberg, Elisabet; Loftenius, Annika; Frejd, Fredrik Y; Tolmachev, Vladimir

Novel Chlorin with a HYNIC: Synthesis, (99m)Tc-Radiolabeling, and Initial Preclinical Evaluation

新型含HYNIC基团的氯化合物:合成、(99m)Tc放射性标记及初步临床前评价

Popov, Alexander; Suvorov, Nikita; Larkina, Mariia; Plotnikov, Evgenii; Varvashenya, Ruslan; Bodenko, Vitalina; Yanovich, Gleb; Ostroverkhov, Petr; Usachev, Maxim; Filonenko, Elena; Belousov, Mikhail; Grin, Mikhail

Synthesis and Preclinical Evaluation of Urea-Based Prostate-Specific Membrane Antigen-Targeted Conjugates Labeled with (177)Lu

尿素基前列腺特异性膜抗原靶向缀合物(177Lu标记)的合成及临床前评价

Machulkin, Aleksei E; Petrov, Stanislav A; Bodenko, Vitalina; Larkina, Mariia S; Plotnikov, Evgenii; Yuldasheva, Feruza; Tretyakova, Maria; Bezverkhniaia, Ekaterina; Zyk, Nikolay Yu; Stasyuk, Elena; Zelchan, Roman; Majouga, Alexander G; Tolmachev, Vladimir; Orlova, Anna; Beloglazkina, Elena K; Yusubov, Mekhman S

(177)Lu-labeled PSMA targeting therapeutic with optimized linker for treatment of disseminated prostate cancer; evaluation of biodistribution and dosimetry

(177)Lu标记的PSMA靶向治疗药物,采用优化的连接子治疗转移性前列腺癌;生物分布和剂量学评价

Abouzayed, Ayman; Seitova, Kamila; Lundmark, Fanny; Bodenko, Vitalina; Oroujeni, Maryam; Tolmachev, Vladimir; Rosenström, Ulrika; Orlova, Anna

Visualization of epithelial cell adhesion molecule-expressing renal cell carcinoma xenografts using designed ankyrin repeat protein Ec1 labelled with (99m)Tc and (125)I

利用经设计的锚蛋白重复序列蛋白 Ec1 标记(99mTc 和 125I),对表达上皮细胞黏附分子的肾细胞癌异种移植瘤进行可视化。

Tolmachev, Vladimir; Bodenko, Vitalina; Orlova, Anna; Schulga, Alexey; Deyev, Sergey M; Vorobyeva, Anzhelika

Synthesis, 123I-Radiolabeling Optimization, and Initial Preclinical Evaluation of Novel Urea-Based PSMA Inhibitors with a Tributylstannyl Prosthetic Group in Their Structures

结构中含有三丁基锡烷基辅基的新型尿素基 PSMA 抑制剂的合成、123I 放射性标记优化及初步临床前评估

Lutfi A Hasnowo, Maria S Larkina, Evgenii Plotnikov, Vitalina Bodenko, Feruza Yuldasheva, Elena Stasyuk, Stanislav A Petrov, Nikolai Y Zyk, Aleksei E Machulkin, Nikolai I Vorozhtsov, Elena K Beloglazkina, Valentine G Nenajdenko, Vladimir Tolmachev, Anna Orlova, Alexander G Majouga, Mekhman S Yusubov

Preclinical Evaluation of a New Format of (68)Ga- and (111)In-Labeled Affibody Molecule Z(IGF-1R:4551) for the Visualization of IGF-1R Expression in Malignant Tumors Using PET and SPECT

利用PET和SPECT对新型(68)Ga和(111)In标记的Affibody分子Z(IGF-1R:4551)进行临床前评估,用于可视化恶性肿瘤中IGF-1R的表达。

Liu, Yongsheng; Yu, Shengze; Xu, Tianqi; Bodenko, Vitalina; Orlova, Anna; Oroujeni, Maryam; Rinne, Sara S; Tolmachev, Vladimir; Vorobyeva, Anzhelika; Gräslund, Torbjörn

Biologic Evaluation of a Heterodimeric HER2-Albumin Targeted Affibody Molecule Produced by Chemo-Enzymatic Peptide Synthesis

化学酶肽合成产生的异二聚 HER2-白蛋白靶向 Affibody 分子的生物学评价

Yongsheng Liu, Rezan Güler, Yunqi Liao, Anzhelika Vorobyeva, Olof Widmark, Theodorus J Meuleman, Anna Koijen, Leendert J van den Bos, Robert Naasz, Vitalina Bodenko, Anna Orlova, Caroline Ekblad, Vladimir Tolmachev, Fredrik Y Frejd

Effect of Inter-Domain Linker Composition on Biodistribution of ABD-Fused Affibody-Drug Conjugates Targeting HER2

域间接头组成对针对 HER2 的 ABD 融合 Affibody-药物偶联物的生物分布的影响

Tianqi Xu, Jie Zhang, Maryam Oroujeni, Maria S Tretyakova, Vitalina Bodenko, Mikhail V Belousov, Anna Orlova, Vladimir Tolmachev, Anzhelika Vorobyeva, Torbjörn Gräslund