日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Biphenyl as a Privileged Structure in Medicinal Chemistry: Advances in Anti-Infective Drug Discovery

联苯作为药物化学中的优势结构:抗感染药物发现的进展

Gandi, Marilia Oliva; França, Rodolfo Rodrigo Florido; Castelo-Branco, Frederico Silva; Boechat, Nubia

Discovery of [1,2,4]triazolo[1,5-a]pyrimidine-Imatinib Hybrids With Selective Cytotoxic Activity: A Mechanistically Divergent Series From Direct BCR-ABL1 Inhibition

发现具有选择性细胞毒活性的[1,2,4]三唑并[1,5-a]嘧啶-伊马替尼杂合物:与直接抑制BCR-ABL1机制不同的系列

Moura, Stefany Castro Bazan; de Oliveira, Andressa Paula; Neto, Joao de Mello Rezende; Dantas, Rafael Ferreira; Silva-Jr, Floriano Paes; Pimentel, Luiz Claudio; Carvalho, Mayara Salles do Nascimento; Leite, Debora Inacio; da Silva, Daiane Vitoria; Bastos, Monica Macedo; Boechat, Nubia

Antiviral Activity of Pyrazolopyrimidine and Triazolopyrimidine Derivatives Against SARS-CoV-2 In Vitro: Identifying PZP25 as a Promising Scaffold

吡唑并嘧啶和三唑并嘧啶衍生物对SARS-CoV-2的体外抗病毒活性:鉴定PZP25为有前景的骨架

Sardar, Saiqa; Martins, Jessica S C C; Sousa, Thiago C; Silva, Andreon S M; Pinto, Marcelo A; Silveira, Flávia F; Silva, Thais B; França, Rodolfo R F; Pinheiro, Luiz C S; Boechat, Nubia; Siqueira, Marilda M; Matos, Aline R; Carvalho, Leonardo J M

A Review on Medicinal Chemistry and Biological Activity of Dihydropyrimidinones Against HIV

二氢嘧啶酮类药物的药物化学及抗HIV生物活性研究综述

Leite, Debora I; Macedo, Fernando B; Lima, Murilo Marinho de C; Brum, Isabelle S; Oliveira, Jonathan Fragoso Miranda de; Costa, Ana Clara S; Duarte, Stella C; Moon, Sarah; Moura, Stefany de Castro B; Oliveira, Andressa P de; Boechat, Nubia; Bastos, Monica M

Molluscicidal and Schistosomicidal Activities of 2-(1H-Pyrazol-1-yl)-1,3,4-thiadiazole Derivatives

2-(1H-吡唑-1-基)-1,3,4-噻二唑衍生物的杀软体动物和杀血吸虫活性

da Silva Rangel, Leonardo; Gonzaga, Daniel Tadeu Gomes; da Silva, Ana Cláudia Rodrigues; von Ranke, Natalia Lindmar; Rodrigues, Carlos Rangel; Santos, José Augusto Albuquerque Dos; Boechat, Nubia; Gomes, Keyla Nunes Farias; Teixeira, Guilherme Pegas; Faria, Robson Xavier

Design, Synthesis, and Biological Evaluation of N-Acylhydrazones and Their Activity Against Leishmania amazonensis Promastigotes

N-酰基腙的设计、合成及生物学评价及其对亚马逊利什曼原虫前鞭毛体的活性

Oliveira Monteiro, Caio Eduardo; Martins Mafra, João Carlos; Boechat, Nubia; Silva, Edson Roberto da

Ponatinib: A Review of the History of Medicinal Chemistry behind Its Development

帕纳替尼:其研发背后的药物化学史回顾

Nascimento, Mayara; Moura, Stefany; Parra, Lidia; Vasconcellos, Valeska; Costa, Gabriela; Leite, Debora; Dias, Maria; Fernandes, Tácio Vinício Amorim; Hoelz, Lucas; Pimentel, Luiz; Bastos, Monica; Boechat, Nubia

A Review of the Development of Multitarget Molecules against HIV-TB Coinfection Pathogens

针对HIV-TB合并感染病原体的多靶点分子研发进展综述

Leite, Debora Inacio; de Castro Bazan Moura, Stefany; da Conceição Avelino Dias, Maria; Costa, Carolina Catta Preta; Machado, Gustavo Peixoto; Pimentel, Luiz Claudio Ferreira; Branco, Frederico Silva Castelo; Moreira, Rui; Bastos, Monica Macedo; Boechat, Nubia

The Use of Zidovudine Pharmacophore in Multi-Target-Directed Ligands for AIDS Therapy

齐多夫定药效团在多靶点导向配体治疗艾滋病中的应用

Bianco, Maria da Conceição Avelino Dias; Inacio Leite, Debora; Silva Castelo Branco, Frederico; Boechat, Nubia; Uliassi, Elisa; Bolognesi, Maria Laura; Bastos, Monica Macedo

New Imatinib Derivatives with Antiproliferative Activity against A549 and K562 Cancer Cells.

具有抗A549和K562癌细胞增殖活性的新型伊马替尼衍生物

Oliveira Andressa, Moura Stefany, Pimentel Luiz, Neto João, Dantas Rafael, Silva-Jr Floriano, Bastos Monica, Boechat Nubia