日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

GTP release-selective agonists prolong opioid analgesic efficacy

GTP释放选择性激动剂可延长阿片类镇痛药的疗效。

Stahl, Edward L; Swanson, Matthew A; Dang, Vuong Q; Cameron, Michael D; Kennedy, Nicole M; Bannister, Thomas D; Bohn, Laura M

Crystal structures of agonist-bound human cannabinoid receptor CB(1)

激动剂结合的人类大麻素受体CB(1)的晶体结构

Hua, Tian; Vemuri, Kiran; Nikas, Spyros P; Wu, Yiran; Qu, Lu; Pu, Mengchen; Korde, Anisha; Jiang, Shan; Ho, Jo-Hao; Han, Gye Won; Ding, Kang; Li, Xuanxuan; Liu, Haiguang; Hanson, Michael A; Zhao, Suwen; Bohn, Laura M; Makriyannis, Alexandros; Stevens, Raymond C; Liu, Zhi-Jie

Retraction Note: Crystal structures of agonist-bound human cannabinoid receptor CB(1)

撤稿声明:激动剂结合的人类大麻素受体 CB(1) 的晶体结构

Hua, Tian; Vemuri, Kiran; Nikas, Spyros P; Laprairie, Robert B; Wu, Yiran; Qu, Lu; Pu, Mengchen; Korde, Anisha; Jiang, Shan; Ho, Jo-Hao; Han, Gye Won; Ding, Kang; Li, Xuanxuan; Liu, Haiguang; Hanson, Michael A; Zhao, Suwen; Bohn, Laura M; Makriyannis, Alexandros; Stevens, Raymond C; Liu, Zhi-Jie

Characterization of the GTPγS release function of a G protein-coupled receptor

对G蛋白偶联受体的GTPγS释放功能进行表征

Bohn, Laura M; Stahl, Edward L

Bidirectional Modification of a Galbulimima Alkaloid Identifies Selective Opioid Ligands

Galbulimima 生物碱的双向修饰可鉴定选择性阿片类配体

Zielke, Florian Martin; Woo, Stone; Kasmali, Samuel; Volf, Allison; Dang, Vuong Q; Bailey, Jake B; Gembicky, Milan; Bohn, Laura M; Shenvi, Ryan A

Exceptionally Potent Chiral Anandamide Analogs.

超强效手性花生四烯酸乙醇胺类似物。

Georgiadis Markos-Orestis, Ferreras Elena, Ji Lipin, Ferreira Luana Assis, Hainline John, Tong Fei, Dang Vuong Q, Faragher Alexandra, Sadybekov Anastasiia V, Bohn Laura M, Katritch Vsevolod, Hohmann Andrea G, Makriyannis Alexandros, Nikas Spyros P

Novel Tetraolefinic Chain Phenyl Substituted Endocannabinoid Probes.

新型四烯烃链苯基取代内源性大麻素探针。

Georgiadis Markos-Orestis, Ji Lipin, Tong Fei, Dang Vuong Q, Ferreira Luana Assis, Faragher Alexandra, Tran Ngan, Sadybekov Anastasiia V, Ganapathy Suthakar, Zvonok Nikolai, Katritch Vsevolod, Hohmann Andrea G, Bohn Laura M, Makriyannis Alexandros, Nikas Spyros P

Depression of intracranial self-stimulation in male and female rats by intraperitoneal lactic acid: effects of morphine, ketoprofen, and interactions with G-protein biased kappa opioid agonists

腹腔注射乳酸抑制雄性和雌性大鼠颅内自刺激:吗啡、酮洛芬的作用以及与G蛋白偏向性κ阿片受体激动剂的相互作用

Martin, Thomas J; Martin, Conner W; Frankowski, Kevin J; Blough, Bruce E; Aubé, Jeffrey; Bohn, Laura M; Jones, Sara R

Triazole 187 is a biased KOR agonist that suppresses itch without sedation and induces anxiolytic-like behaviors in mice

三唑187是一种偏向性κ阿片受体激动剂,可在不引起镇静的情况下抑制瘙痒,并诱导小鼠产生类似抗焦虑的行为。

Volf, Allison; Brust, Tarsis F; Kobylski, Robin R; Czekner, Kerri M; Stahl, Edward L; Cameron, Michael D; Trojniak, Ashley E; Aubé, Jeffrey; Bohn, Laura M

Comparison of Agonist Activity between CB1 and CB2 Receptors with Orthosteric Site Mutations

CB1和CB2受体正构位点突变激动剂活性的比较

Brust, Christina A; Swanson, Matthew A; Iliopoulos Tsoutsouvas, Christos; Dimova, Snezana T; Dang, Vuong Q; Stahl, Edward L; Ho, Jo-Hao; Nikas, Spyros P; Makriyannis, Alexandros; Bohn, Laura M