日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a novel small molecule degrader of wild type and mutant estrogen receptors using DNA encoded libraries

利用DNA编码文库发现一种新型小分子降解剂,可降解野生型和突变型雌激素受体。

Devakrishnan, Anil Kumar; Madasu, Chandrashekhar; Wang, Yong; Modukuri, Ramkumar; Bohren, Kurt M; MacKenzie, Kevin R; Young, Damian W; Fuqua, Suzanne A W; Matzuk, Martin M; Palaniappan, Murugesan

Reversible male contraception by targeted inhibition of serine/threonine kinase 33

通过靶向抑制丝氨酸/苏氨酸激酶33实现可逆性男性避孕

Ku, Angela F; Sharma, Kiran L; Ta, Hai Minh; Sutton, Courtney M; Bohren, Kurt M; Wang, Yong; Chamakuri, Srinivas; Chen, Ruihong; Hakenjos, John M; Jimmidi, Ravikumar; Kent, Katarzyna; Li, Feng; Li, Jian-Yuan; Ma, Lang; Madasu, Chandrashekhar; Palaniappan, Murugesan; Palmer, Stephen S; Qin, Xuan; Robers, Matthew B; Sankaran, Banumathi; Tan, Zhi; Vasquez, Yasmin M; Wang, Jian; Wilkinson, Jennifer; Yu, Zhifeng; Ye, Qiuji; Young, Damian W; Teng, Mingxing; Kim, Choel; Matzuk, Martin M

Discovery of highly potent and ALK2/ALK1 selective kinase inhibitors using DNA-encoded chemistry technology.

利用DNA编码化学技术发现高效且对ALK2/ALK1具有选择性的激酶抑制剂

Jimmidi Ravikumar, Monsivais Diana, Ta Hai Minh, Sharma Kiran L, Bohren Kurt M, Chamakuri Srinivas, Liao Zian, Li Feng, Hakenjos John M, Li Jian-Yuan, Mishina Yuji, Pan Haichun, Qin Xuan, Robers Matthew B, Sankaran Banumathi, Tan Zhi, Tang Suni, Vasquez Yasmin M, Wilkinson Jennifer, Young Damian W, Palmer Stephen S, MacKenzie Kevin R, Kim Choel, Matzuk Martin M

DNA-encoded chemistry technology yields expedient access to SARS-CoV-2 M(pro) inhibitors.

DNA编码化学技术可快速获得SARS-CoV-2 M(pro)抑制剂

Chamakuri Srinivas, Lu Shuo, Ucisik Melek Nihan, Bohren Kurt M, Chen Ying-Chu, Du Huang-Chi, Faver John C, Jimmidi Ravikumar, Li Feng, Li Jian-Yuan, Nyshadham Pranavanand, Palmer Stephen S, Pollet Jeroen, Qin Xuan, Ronca Shannon E, Sankaran Banumathi, Sharma Kiran L, Tan Zhi, Versteeg Leroy, Yu Zhifeng, Matzuk Martin M, Palzkill Timothy, Young Damian W

NELL2-mediated lumicrine signaling through OVCH2 is required for male fertility

NELL2介导的通过OVCH2的泌尿道信号传导是男性生育力所必需的

Kiyozumi, Daiji; Noda, Taichi; Yamaguchi, Ryo; Tobita, Tomohiro; Matsumura, Takafumi; Shimada, Kentaro; Kodani, Mayo; Kohda, Takashi; Fujihara, Yoshitaka; Ozawa, Manabu; Yu, Zhifeng; Miklossy, Gabriella; Bohren, Kurt M; Horie, Masato; Okabe, Masaru; Matzuk, Martin M; Ikawa, Masahito

Discovery of potent thrombin inhibitors from a protease-focused DNA-encoded chemical library

从以蛋白酶为靶点的DNA编码化合物库中发现强效凝血酶抑制剂

Dawadi, Surendra; Simmons, Nicholas; Miklossy, Gabriella; Bohren, Kurt M; Faver, John C; Ucisik, Melek Nihan; Nyshadham, Pranavanand; Yu, Zhifeng; Matzuk, Martin M

C-N Coupling of DNA-Conjugated (Hetero)aryl Bromides and Chlorides for DNA-Encoded Chemical Library Synthesis

DNA偶联(杂)芳基溴化物和氯化物的CN偶联用于DNA编码化学库的合成

Chen, Ying-Chu; Faver, John C; Ku, Angela F; Miklossy, Gabriella; Riehle, Kevin; Bohren, Kurt M; Ucisik, Melek N; Matzuk, Martin M; Yu, Zhifeng; Simmons, Nicholas

Homogeneous and Functional Group Tolerant Ring-Closing Metathesis for DNA-Encoded Chemical Libraries

用于DNA编码化学库的均相和官能团耐受的闭环复分解反应

Monty, Olivier B C; Nyshadham, Pranavanand; Bohren, Kurt M; Palaniappan, Murugesan; Matzuk, Martin M; Young, Damian W; Simmons, Nicholas

Palladium-Catalyzed Hydroxycarbonylation of (Hetero)aryl Halides for DNA-Encoded Chemical Library Synthesis

钯催化(杂)芳基卤化物羟基羰基化反应用于DNA编码化学库的合成

Li, Jian-Yuan; Miklossy, Gabriella; Modukuri, Ram K; Bohren, Kurt M; Yu, Zhifeng; Palaniappan, Murugesan; Faver, John C; Riehle, Kevin; Matzuk, Martin M; Simmons, Nicholas

Arginine Metabolism Is Altered in Adults with A-β + Ketosis-Prone Diabetes

患有A-β+酮症倾向型糖尿病的成年人精氨酸代谢发生改变

Mulukutla, Surya N; Hsu, Jean W; Gaba, Ruchi; Bohren, Kurt M; Guthikonda, Anu; Iyer, Dinakar; Ajami, Nadim J; Petrosino, Joseph F; Hampe, Christiane S; Ram, Nalini; Jahoor, Farook; Balasubramanyam, Ashok