日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Non-clinical and first-in-human characterization of ECC5004/AZD5004, a novel once-daily, oral small-molecule GLP-1 receptor agonist

ECC5004/AZD5004 是一种新型每日一次口服小分子 GLP-1 受体激动剂,对其进行非临床和首次人体表征。

Haggag, Amina Z; Xu, Jianfeng; Butcher, Laurie; Pagnussat, Sandra; Davies, Graeme; Lundqvist, Sara; Wang, Wenyu; Van Zuydam, Natalie; Nelander, Karin; Jha, Aruni; Yu, Hongtao; Boianelli, Alessandro; Lindmark, Bosse; Ollerstam, Anna; Sun, Xuefeng; Wang, Fan; Pan, Xiaoliang; Liu, Haihui; Chen, Wengang; Xu, Jianfeng; Wallenius, Kristina; Zhou, Jingye

Knockdown of ketohexokinase versus inhibition of its kinase activity exert divergent effects on fructose metabolism

敲除酮己糖激酶与抑制其激酶活性对果糖代谢产生截然不同的影响。

Park, Se-Hyung; Fadhul, Taghreed; Conroy, Lindsey R; Clarke, Harrison A; Sun, Ramon C; Wallenius, Kristina; Boucher, Jeremie; O'Mahony, Gavin; Boianelli, Alessandro; Persson, Marie; Jung, Sunhee; Jang, Cholsoon; Loria, Analia S; Martinez, Genesee J; Kipp, Zachary A; Bates, Evelyn A; Hinds, Terry D Jr; Divanovic, Senad; Softic, Samir

Cross-Species Translation of Biophase Half-Life and Potency of GalNAc-Conjugated siRNAs

GalNAc偶联siRNA的生物相半衰期和效力的跨物种翻译

Boianelli, Alessandro; Aoki, Yasunori; Ivanov, Maxim; Dahlén, Anders; Gennemark, Peter

A non-linear deterministic model for regulation of diauxic lag on cellobiose by the pneumococcal multidomain transcriptional regulator CelR.

肺炎球菌多结构域转录调节因子 CelR 对纤维二糖双相滞后期的调控非线性确定性模型

Boianelli Alessandro, Bidossi Alessandro, Gualdi Luciana, Mulas Laura, Mocenni Chiara, Pozzi Gianni, Vicino Antonio, Oggioni Marco R