日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Analysis of Burkholderia pseudomallei IspF in complex with sulfapyridine, sulfamonomethoxine, ethoxzolamide and acetazolamide

分析类鼻疽伯克霍尔德菌 IspF 与磺胺吡啶、磺胺甲氧嘧啶、乙氧唑胺和乙酰唑胺的复合物

Grote, Dakota; Stewart, Christopher G; Daraji, Drashti G; Enayati, Parisa; Braverman, Kristina N; Romanaggi, CeAnn; Bolejack, Madison J; Yano, Jason K; Abendroth, Jan; Dranow, David M; Pierce, Phillip G; Lorimer, Donald D; Horanyi, Peter S; Staker, Bart L; Edwards, Thomas E; Myler, Peter J; Horn, James R; Hagen, Timothy J

Enolase inhibitors as therapeutic leads for Naegleria fowleri infection

烯醇化酶抑制剂作为治疗福氏耐格里阿米巴原虫感染的线索

Jillian E Milanes, Victoria C Yan, Cong-Dat Pham, Florian Muller, Samuel Kwain, Kerrick C Rees, Brian N Dominy, Daniel C Whitehead, Steven W Millward, Madison Bolejack, Roger Shek, Logan Tillery, Isabelle Q Phan, Bart Staker, E Ashley Moseman, Xiang Zhang, Xipeng Ma, Audriy Jebet, Xinmin Yin, James

Crystal structure and biophysical characterization of IspD from Burkholderia thailandensis and Mycobacterium paratuberculosis

泰国伯克霍尔德菌和副结核分枝杆菌IspD的晶体结构和生物物理特性

Pierce, Phillip G; Hartnett, Brian E; Laughlin, Tosha M; Blain, Joy M; Mayclin, Stephen J; Bolejack, Madison J; Myers, Janette B; Higgins, Tate W; Dranow, David M; Sullivan, Amy; Lorimer, Donald D; Edwards, Thomas E; Hagen, Timothy J; Horn, James R; Myler, Peter J

A phase II trial of regorafenib in patients with advanced Ewing sarcoma and related tumors of soft tissue and bone: SARC024 trial results

瑞戈非尼治疗晚期尤文氏肉瘤及相关软组织和骨肿瘤患者的II期临床试验:SARC024试验结果

Attia, Steven; Bolejack, Vanessa; Ganjoo, Kristen N; George, Suzanne; Agulnik, Mark; Rushing, Daniel; Loggers, Elizabeth T; Livingston, Michael B; Wright, Jennifer; Chawla, Sant P; Okuno, Scott H; Reinke, Denise K; Riedel, Richard F; Davis, Lara E; Ryan, Christopher W; Maki, Robert G

Structure-Guided Discovery of N(5)-CAIR Mutase Inhibitors

基于结构的N(5)-CAIR变位酶抑制剂发现

Belfon, Kafi K J; Sharma, Nandini; Zigweid, Rachael; Bolejack, Madison; Davies, Doug; Edwards, Thomas E; Myler, Peter J; French, Jarrod B

Bacterial structural genomics target enabled by a recently discovered potent fungal acetyl-CoA synthetase inhibitor

细菌结构基因组学研究得益于近期发现的一种强效真菌乙酰辅酶A合成酶抑制剂

DeBouver, Nicholas D; Bolejack, Madison J; Esan, Taiwo E; Krysan, Damian J; Hagen, Timothy J; Abendroth, Jan

Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1

发现并表征了一系列新型氯嘧啶类化合物作为激酶 MSK1 的共价抑制剂

Hall, Adrian; Abendroth, Jan; Bolejack, Madison J; Ceska, Tom; Dell'Aiera, Sylvie; Ellis, Victoria; Fox, David 3rd; François, Cyril; Muruthi, Muigai M; Prével, Camille; Poullennec, Karine; Romanov, Sergei; Valade, Anne; Vanbellinghen, Alain; Yano, Jason; Geraerts, Martine

Regulation of multiple dimeric states of E-cadherin by adhesion activating antibodies revealed through Cryo-EM and X-ray crystallography

通过低温电子显微镜和 X 射线晶体学揭示粘附激活抗体对 E-钙粘蛋白多种二聚体状态的调节

Allison Maker, Madison Bolejack, Leslayann Schecterson, Brad Hammerson, Jan Abendroth, Thomas E Edwards, Bart Staker, Peter J Myler, Barry M Gumbiner

TRANSFORMER: A Randomized Phase II Study Comparing Bipolar Androgen Therapy Versus Enzalutamide in Asymptomatic Men With Castration-Resistant Metastatic Prostate Cancer

TRANSFORMER:一项随机II期研究,比较双极雄激素疗法与恩扎卢胺治疗无症状去势抵抗性转移性前列腺癌男性患者的疗效

Denmeade, Samuel R; Wang, Hao; Agarwal, Neeraj; Smith, David C; Schweizer, Michael T; Stein, Mark N; Assikis, Vasileios; Twardowski, Przemyslaw W; Flaig, Thomas W; Szmulewitz, Russell Z; Holzbeierlein, Jeffrey M; Hauke, Ralph J; Sonpavde, Guru; Garcia, Jorge A; Hussain, Arif; Sartor, Oliver; Mao, Shifeng; Cao, Harry; Fu, Wei; Wang, Ting; Abdallah, Rehab; Lim, Su Jin; Bolejack, Vanessa; Paller, Channing J; Carducci, Michael A; Markowski, Mark C; Eisenberger, Mario A; Antonarakis, Emmanuel S

Naegleria fowleri: Protein structures to facilitate drug discovery for the deadly, pathogenic free-living amoeba

福氏耐格里阿米巴:蛋白质结构有助于发现针对这种致命致病性自由生活变形虫的药物

Tillery, Logan; Barrett, Kayleigh; Goldstein, Jenna; Lassner, Jared W; Osterhout, Bram; Tran, Nathan L; Xu, Lily; Young, Ryan M; Craig, Justin; Chun, Ian; Dranow, David M; Abendroth, Jan; Delker, Silvia L; Davies, Douglas R; Mayclin, Stephen J; Calhoun, Brandy; Bolejack, Madison J; Staker, Bart; Subramanian, Sandhya; Phan, Isabelle; Lorimer, Donald D; Myler, Peter J; Edwards, Thomas E; Kyle, Dennis E; Rice, Christopher A; Morris, James C; Leahy, James W; Manetsch, Roman; Barrett, Lynn K; Smith, Craig L; Van Voorhis, Wesley C