日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of 7,9-Dibromo-dihydrodibenzofuran as a Potent Casein Kinase 2 (CK2) Inhibitor: Synthesis, Biological Evaluation, and Structural Studies on E-/Z-Isomers.

发现 7,9-二溴二氢二苯并呋喃是一种有效的酪蛋白激酶 2 (CK2) 抑制剂:E-/Z-异构体的合成、生物学评价和结构研究

Rumler Hendrik, Schmithals Claudia, Werner Christian, Bollacke Andre, Aichele Dagmar, Götz Claudia, Niefind Karsten, Wünsch Bernhard, Jose Joachim

Self-Assembled Supramolecular Nanoparticles Improve the Cytotoxic Efficacy of CK2 Inhibitor THN7

自组装超分子纳米粒子提高了CK2抑制剂THN7的细胞毒性功效

Nacereddine, Abdelhamid; Bollacke, Andre; Róka, Eszter; Marminon, Christelle; Bouaziz, Zouhair; Fenyvesi, Ferenc; Bácskay, Ildikó Katalin; Jose, Joachim; Perret, Florent; Le Borgne, Marc

Identification of a Potent Allosteric Inhibitor of Human Protein Kinase CK2 by Bacterial Surface Display Library Screening

利用细菌表面展示文库筛选鉴定人蛋白激酶CK2的强效变构抑制剂

Nienberg, Christian; Garmann, Claudia; Gratz, Andreas; Bollacke, Andre; Götz, Claudia; Jose, Joachim

Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity

酚类茚并[1,2-b]吲哚类化合物作为ABCG2选择性强效无毒抑制剂,可刺激基础ATPase活性

Gozzi, Gustavo Jabor; Bouaziz, Zouhair; Winter, Evelyn; Daflon-Yunes, Nathalia; Honorat, Mylène; Guragossian, Nathalie; Marminon, Christelle; Valdameri, Glaucio; Bollacke, Andre; Guillon, Jean; Pinaud, Noël; Marchivie, Mathieu; Cadena, Silvia M; Jose, Joachim; Le Borgne, Marc; Di Pietro, Attilio

Functional display of heterotetrameric human protein kinase CK2 on Escherichia coli: a novel tool for drug discovery

在大肠杆菌上功能性展示异源四聚体人蛋白激酶CK2:一种新型药物发现工具

Gratz, Andreas; Bollacke, Andre; Stephan, Sara; Nienberg, Christian; Le Borgne, Marc; Götz, Claudia; Jose, Joachim

Synthesis, Biological Evaluation and Molecular Modeling of Substituted Indeno[1,2-b]indoles as Inhibitors of Human Protein Kinase CK2

取代的茚并[1,2-b]吲哚类化合物作为人蛋白激酶CK2抑制剂的合成、生物学评价和分子建模

Alchab, Faten; Ettouati, Laurent; Bouaziz, Zouhair; Bollacke, Andre; Delcros, Jean-Guy; Gertzen, Christoph G W; Gohlke, Holger; Pinaud, Noël; Marchivie, Mathieu; Guillon, Jean; Fenet, Bernard; Jose, Joachim; Borgne, Marc Le