日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

CREBBP/EP300 acetyltransferase inhibition disrupts FOXA1-bound enhancers to inhibit the proliferation of ER+ breast cancer cells

CREBBP/EP300 乙酰转移酶抑制可破坏 FOXA1 结合增强子，从而抑制 ER+ 乳腺癌细胞的增殖

期刊:PLoS One
影响因子:2.9
doi:10.1371/journal.pone.0262378
Archana Bommi-Reddy, Sungmi Park-Chouinard, David N Mayhew, Esteban Terzo, Aparna Hingway, Michael J Steinbaugh, Jonathan E Wilson, Robert J Sims 3rd, Andrew R Conery
肿瘤
乳腺癌
肿瘤细胞
WB
发表日期：2022
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Discovery of CPI-1612: A Potent, Selective, and Orally Bioavailable EP300/CBP Histone Acetyltransferase Inhibitor

CPI-1612 的发现：一种高效、选择性强且口服生物利用度高的 EP300/CBP 组蛋白乙酰转移酶抑制剂

期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.0c00155
Wilson, Jonathan E; Patel, Gaurav; Patel, Chirag; Brucelle, Francois; Huhn, Annissa; Gardberg, Anna S; Poy, Florence; Cantone, Nico; Bommi-Reddy, Archana; Sims, Robert J 3rd; Cummings, Richard T; Levell, Julian R
EP300
P300
CBP
发表日期：2020
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Bromodomain inhibition of the transcriptional coactivators CBP/EP300 as a therapeutic strategy to target the IRF4 network in multiple myeloma

转录辅激活因子 CBP/EP300 的溴结构域抑制作为针对多发性骨髓瘤 IRF4 网络的治疗策略

期刊:Elife
影响因子:6.4
doi:10.7554/eLife.10483
Andrew R Conery, Richard C Centore, Adrianne Neiss, Patricia J Keller, Shivangi Joshi, Kerry L Spillane, Peter Sandy, Charlie Hatton, Eneida Pardo, Laura Zawadzke, Archana Bommi-Reddy, Karen E Gascoigne, Barbara M Bryant, Jennifer A Mertz, Robert J Sims
肿瘤
骨髓瘤
WB
发表日期：2016
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Correction: Bromodomain inhibition of the transcriptional coactivators CBP/EP300 as a therapeutic strategy to target the IRF4 network in multiple myeloma

更正：溴结构域抑制转录共激活因子CBP/EP300作为靶向多发性骨髓瘤中IRF4网络的治疗策略

期刊:Elife
影响因子:6.4
doi:10.7554/eLife.19432
Conery, Andrew R; Centore, Richard C; Neiss, Adrianne; Keller, Patricia J; Joshi, Shivangi; Spillane, Kerry L; Sandy, Peter; Hatton, Charlie; Pardo, Eneida; Zawadzke, Laura; Bommi-Reddy, Archana; Gascoigne, Karen E; Bryant, Barbara M; Mertz, Jennifer A; Sims, Robert J
P300
多发性骨髓瘤
CBP
EP300
骨髓瘤
发表日期：2016
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Kinase requirements in human cells: III. Altered kinase requirements in VHL-/- cancer cells detected in a pilot synthetic lethal screen

人类细胞中的激酶需求：III. 在初步合成致死筛选中检测到的VHL-/-癌细胞中激酶需求的改变

期刊:Proceedings of the National Academy of Sciences of the United States of America
影响因子:9.1
doi:10.1073/pnas.0806574105
Bommi-Reddy, Archana; Almeciga, Ingrid; Sawyer, Jacqueline; Geisen, Christoph; Li, Wenliang; Harlow, Ed; Kaelin, William G Jr; Grueneberg, Dorre A
肿瘤
肿瘤免疫
信号转导
细胞生物学
VHL
发表日期：2008
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