日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer.

基于结构的Hsp90/HDAC6双重抑制剂的发现及其在侵袭性前列腺癌中的应用

Citarella Andrea, Belluti Silvia, Bonanni Davide, Moi Davide, Piccinini Isabella, Rinaldi Arianna, Papulino Chiara, Benedetti Rosaria, Cuoghi Laura, Ciolo Stefano Di, Silvani Alessandra, Altucci Lucia, Pinzi Luca, Franchini Silvia, Passarella Daniele, Sorbi Claudia, Giannini Clelia, Imbriano Carol, Rastelli Giulio

Development of machine learning classifiers to predict compound activity on prostate cancer cell lines

开发机器学习分类器以预测化合物对前列腺癌细胞系的活性

Bonanni, Davide; Pinzi, Luca; Rastelli, Giulio

Hydroxamic Acid Derivatives: From Synthetic Strategies to Medicinal Chemistry Applications

羟肟酸衍生物:从合成策略到药物化学应用

Citarella, Andrea; Moi, Davide; Pinzi, Luca; Bonanni, Davide; Rastelli, Giulio

Exploration of [2 + 2 + 2] cyclotrimerisation methodology to prepare tetrahydroisoquinoline-based compounds with potential aldo-keto reductase 1C3 target affinity

探索[2 + 2 + 2]环三聚反应方法制备具有潜在醛酮还原酶1C3靶向亲和力的四氢异喹啉类化合物。

Santos, Ana R N; Sheldrake, Helen M; Ibrahim, Ali I M; Danta, Chhanda Charan; Bonanni, Davide; Daga, Martina; Oliaro-Bosso, Simonetta; Boschi, Donatella; Lolli, Marco L; Pors, Klaus