日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

Inhibiting microtubule polymerization with EAPB02303, a prodrug activated by catechol-O-methyl transferase, enhances paclitaxel effect in pancreatic cancer models

EAPB02303是一种由儿茶酚-O-甲基转移酶激活的前药，它能抑制微管聚合，从而增强紫杉醇在胰腺癌模型中的疗效。

期刊:Cell Death & Disease
影响因子:9.6
doi:10.1038/s41419-025-07747-1
Bigot, Kévin; Patinote, Cindy; Garambois, Véronique; Chouchou, Adrien; Gayraud-Paniagua, Stéphanie; Vie, Nadia; Maggipinto, Yann; Smyej, Elias; Robin, Mathilde; Machu, Margot; Bruciamacchie, Marine; Colombo, Pierre-Emmanuel; Bousquet, Corinne; Mathonnet, Muriel; Levy-Augé, Ela; Tosi, Diego; Bonnet, Pierre-Antoine; Gongora, Céline; Deleuze-Masquéfa, Carine; Larbouret, Christel
胰腺癌
肿瘤
肿瘤免疫
发表日期：2025
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The Novel Imiqualine EAPB02303 Is a Potent Drug for Treating Acute Myeloid Leukemia.

新型咪喹啉 EAPB02303 是一种治疗急性髓系白血病的强效药物

期刊:Biomolecules
影响因子:4.8
doi:10.3390/biom15050741
Makhoul Perla, Hleihel Rita, Itani Shaymaa, Hamie Maguy, Pagniagua-Gayraud Stephanie, Patinote Cindy, Richaud Myriam, Merhi Raghida Abou, El-Sabban Marwan, Galas Simon, Deleuze-Masquefa Carine, Bonnet Pierre-Antoine, El Hajj Hiba
肿瘤
白血病
发表日期：2025
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Research Progress on the Structure-activity Relationship and Mechanism of Flavonoid Derivatives in the Treatment of Lung Cancer

黄酮类衍生物治疗肺癌的构效关系及机制研究进展

期刊:Molecules
影响因子:4.6
doi:10.3390/molecules30081827
Yao, Jiacheng; Zhu, Feng; Feng, Yikun; Gu, Chen; Wang, Tianyu; Li, Xinyu; Yang, Hao; Hu, Xiamin; Bonnet, Pierre-Antoine; Meng, Xiangguo
肺癌
肿瘤
肿瘤免疫
发表日期：2025
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Uncovering the Molecular Pathways Implicated in the Anti-Cancer Activity of the Imidazoquinoxaline Derivative EAPB02303 Using a Caenorhabditis elegans Model

利用秀丽隐杆线虫模型揭示咪唑喹喔啉衍生物EAPB02303抗癌活性相关的分子通路

期刊:International Journal of Molecular Sciences
影响因子:4.9
doi:10.3390/ijms25147785
Makhoul, Perla; Galas, Simon; Paniagua-Gayraud, Stéphanie; Deleuze-Masquefa, Carine; Hajj, Hiba El; Bonnet, Pierre-Antoine; Richaud, Myriam
C. elegans
发表日期：2024
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Imiquimod Reverses Chronic Toxoplasmosis-Associated Behavioral and Neurocognitive Anomalies in a Rat Model.

咪喹莫特可逆转大鼠模型中慢性弓形虫病相关的行为和神经认知异常

期刊:Biomedicines
影响因子:3.9
doi:10.3390/biomedicines12061295
Itani Shaymaa, Hamie Maguy, El Jammal Reem, Abdine Wassim, Doumit Mark, Charafeddine Adib, El-Sabban Marwan, Patinote Cindy, Masquefa Carine, Bonnet Pierre-Antoine, Obeid Makram, El Hajj Hiba
神经科学
Rat
发表日期：2024
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Recent Advances on Small-Molecule Antagonists Targeting TLR7

靶向TLR7的小分子拮抗剂的最新进展

期刊:Molecules
影响因子:4.6
doi:10.3390/molecules28020634
Zheng, Haoyang; Wu, Peiyang; Bonnet, Pierre-Antoine
TLR7
发表日期：2023
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[1,2,4]triazolo[4,3-a]quinoxaline as Novel Scaffold in the Imiqualines Family: Candidates with Cytotoxic Activities on Melanoma Cell Lines

[1,2,4]三唑并[4,3-a]喹喔啉作为咪唑啉家族的新型骨架：对黑色素瘤细胞系具有细胞毒活性的候选化合物

期刊:Molecules
影响因子:4.6
doi:10.3390/molecules28145478
Patinote, Cindy; Raevens, Sandy; Baumann, Amélie; Pellegrin, Eloise; Bonnet, Pierre-Antoine; Deleuze-Masquéfa, Carine
黑色素瘤
细胞生物学
发表日期：2023
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Agonist and antagonist ligands of toll-like receptors 7 and 8: Ingenious tools for therapeutic purposes

Toll样受体7和8的激动剂和拮抗剂配体：用于治疗目的的巧妙工具

期刊:European Journal of Medicinal Chemistry
影响因子:5.9
doi:10.1016/j.ejmech.2020.112238
Patinote, Cindy; Karroum, Nour Bou; Moarbess, Georges; Cirnat, Natalina; Kassab, Issam; Bonnet, Pierre-Antoine; Deleuze-Masquéfa, Carine
信号转导
发表日期：2020
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Imidazo[1,2-a]quinoxalines Derivatives Grafted with Amino Acids: Synthesis and Evaluation on A375 Melanoma Cells

咪唑并[1,2-a]喹喔啉衍生物与氨基酸接枝：合成及在A375黑色素瘤细胞上的评价

期刊:Molecules
影响因子:4.6
doi:10.3390/molecules23112987
Chouchou, Adrien; Patinote, Cindy; Cuq, Pierre; Bonnet, Pierre-Antoine; Deleuze-Masquéfa, Carine
细胞生物学
黑色素瘤
发表日期：2018
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