Proteomic and Phosphoproteomic Analysis Reveals that Neurokinin-1 Receptor (NK1R) Blockade with Aprepitant in Human Keratinocytes Activates a Distinct Subdomain of EGFR Signaling: Implications for the Anti-Pruritic Activity of NK1R Antagonists
蛋白质组学和磷酸化蛋白质组学分析表明,人类角质形成细胞中的神经激肽 1 受体 (NK1R) 阻断剂阿瑞吡坦可激活 EGFR 信号传导的一个独特子域:对 NK1R 拮抗剂止痒活性的影响
期刊:Medicines
影响因子:
doi:10.3390/medicines6040114
Shawn G Kwatra, Emily Boozalis, Amy H Huang, Cory Nanni, Raveena Khanna, Kyle A Williams, Yevgeniy R Semenov, Callie M Roberts, Robert F Burns, Madison Krischak, Madan M Kwatra
信号转导
神经
表观遗传
其它细胞
Epigenetics
Neuroscience
Human