日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeted β(-)-Particle Plus Conversion and Auger-Electron Therapy with (161)Tb-Labeled Somatostatin Receptor Antagonist DOTA-LM3: A Phase 0 Study

使用 (161)Tb 标记的生长抑素受体拮抗剂 DOTA-LM3 进行靶向 β(-) 粒子增强转化和俄歇电子疗法:一项 0 期研究

Fricke, Julia G; Westerbergh, Frida; McDougall, Lisa; Favaretto, Chiara; Christ, Emanuel; Nicolas, Guillaume P; Geistlich, Susanne; Schmid, David E; Borgna, Francesca; Fani, Melpomeni; Bernhardt, Peter; van der Meulen, Nicholas P; Müller, Cristina; Schibli, Roger; Wild, Damian

First-in-human administration of terbium-161-labelled somatostatin receptor subtype 2 antagonist ([(161)Tb]Tb-DOTA-LM3) in a patient with a metastatic neuroendocrine tumour of the ileum

首次在人体中应用铽-161标记的生长抑素受体2亚型拮抗剂([(161)Tb]Tb-DOTA-LM3)治疗回肠转移性神经内分泌肿瘤患者

Fricke, Julia; Westerbergh, Frida; McDougall, Lisa; Favaretto, Chiara; Christ, Emanuel; Nicolas, Guillaume P; Geistlich, Susanne; Borgna, Francesca; Fani, Melpomeni; Bernhardt, Peter; van der Meulen, Nicholas P; Müller, Cristina; Schibli, Roger; Wild, Damian

Design and Preclinical Evaluation of a Novel Prostate-Specific Membrane Antigen Radioligand Modified with a Transthyretin Binder.

设计和临床前评估一种新型前列腺特异性膜抗原放射性配体,该配体经转甲状腺素结合剂修饰

Vaccarin Christian, Mapanao Ana Katrina, Deberle Luisa M, Becker Anna E, Borgna Francesca, Marzaro Giovanni, Schibli Roger, Müller Cristina

Impact of the mouse model and molar amount of injected ligand on the tissue distribution profile of PSMA radioligands

小鼠模型和注射配体的摩尔量对PSMA放射性配体组织分布的影响

Tschan, Viviane J; Borgna, Francesca; Schibli, Roger; Müller, Cristina

Combination of terbium-161 with somatostatin receptor antagonists-a potential paradigm shift for the treatment of neuroendocrine neoplasms

铽-161与生长抑素受体拮抗剂联合应用——神经内分泌肿瘤治疗的潜在范式转变

Borgna, Francesca; Haller, Stephanie; Rodriguez, Josep M Monné; Ginj, Mihaela; Grundler, Pascal V; Zeevaart, Jan Rijn; Köster, Ulli; Schibli, Roger; van der Meulen, Nicholas P; Müller, Cristina

Preclinical investigations using [(177)Lu]Lu-Ibu-DAB-PSMA toward its clinical translation for radioligand therapy of prostate cancer

利用[(177)Lu]Lu-Ibu-DAB-PSMA进行临床前研究,以期将其转化为前列腺癌放射性配体疗法。

Tschan, Viviane J; Borgna, Francesca; Busslinger, Sarah D; Stirn, Martina; Rodriguez, Josep M Monné; Bernhardt, Peter; Schibli, Roger; Müller, Cristina

Simultaneous Visualization of (161)Tb- and (177)Lu-Labeled Somatostatin Analogues Using Dual-Isotope SPECT Imaging

利用双同位素SPECT成像技术同时可视化(161)Tb和(177)Lu标记的生长抑素类似物

Borgna, Francesca; Barritt, Patrick; Grundler, Pascal V; Talip, Zeynep; Cohrs, Susan; Zeevaart, Jan Rijn; Köster, Ulli; Schibli, Roger; van der Meulen, Nicholas P; Müller, Cristina

Production of Mass-Separated Erbium-169 Towards the First Preclinical in vitro Investigations

大规模分离制备铒-169:迈向首次临床前体外研究

Talip, Zeynep; Borgna, Francesca; Müller, Cristina; Ulrich, Jiri; Duchemin, Charlotte; Ramos, Joao P; Stora, Thierry; Köster, Ulli; Nedjadi, Youcef; Gadelshin, Vadim; Fedosseev, Valentin N; Juget, Frederic; Bailat, Claude; Fankhauser, Adelheid; Wilkins, Shane G; Lambert, Laura; Marsh, Bruce; Fedorov, Dmitry; Chevallay, Eric; Fernier, Pascal; Schibli, Roger; van der Meulen, Nicholas P

Development of a new class of PSMA radioligands comprising ibuprofen as an albumin-binding entity

开发一类新型PSMA放射性配体,该配体包含布洛芬作为白蛋白结合实体

Deberle, Luisa M; Benešová, Martina; Umbricht, Christoph A; Borgna, Francesca; Büchler, Manuel; Zhernosekov, Konstantin; Schibli, Roger; Müller, Cristina

Albumin-Binding PSMA Radioligands: Impact of Minimal Structural Changes on the Tissue Distribution Profile

白蛋白结合PSMA放射性配体:微小结构变化对组织分布的影响

Deberle, Luisa M; Tschan, Viviane J; Borgna, Francesca; Sozzi-Guo, Fan; Bernhardt, Peter; Schibli, Roger; Müller, Cristina