日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A universal cannabinoid CB1 and CB2 receptor TR-FRET kinetic ligand-binding assay.

一种通用的大麻素 CB1 和 CB2 受体 TR-FRET 动力学配体结合测定法

Borrega-Roman Leire, Hoare Bradley L, Kosar Miroslav, Sarott Roman C, Patej Kacper J, Bouma Jara, Scott-Dennis Morgan, Koers Eline J, Gazzi Thais, Mach Leonard, Barrondo Sergio, Sallés Joan, Guba Wolfgang, Kusznir Eric, Nazaré Marc, Rufer Arne C, Grether Uwe, Heitman Laura H, Carreira Erick M, Sykes David A, Veprintsev Dmitry B

Traffic control: Mechanisms of ligand-specific internalization and intracellular distribution of CCR5

交通控制:CCR5配体特异性内化和细胞内分布的机制

Gu, Siyi; Maurya, Svetlana; Lona, Alexis; Borrega Roman, Leire; Salanga, Catherina; Gonzalez, David J; Kufareva, Irina; Handel, Tracy M

Biased Signaling and Its Role in the Genesis of Short- and Long-Acting β(2)-Adrenoceptor Agonists.

偏向性信号传导及其在短效和长效β2-肾上腺素受体激动剂产生中的作用

Phan Ngan T N, Borrega-Roman Leire, Hoare Bradley L, Harwood Clare R, Geary Natalie, Guba Wolfgang, Han Yongqi, Zenko Vladimirs, Koers Eline J, Rufer Arne C, Grether Uwe, Veprintsev Dmitry B, Sykes David A

Molecular determinants of antagonist interactions with chemokine receptors CCR2 and CCR5

拮抗剂与趋化因子受体CCR2和CCR5相互作用的分子决定因素

Dawson, John R D; Wadman, Grant M; Zhang, Penglie; Tebben, Andrew; Carter, Percy H; Gu, Siyi; Shroka, Thomas; Borrega-Roman, Leire; Salanga, Catherina L; Handel, Tracy M; Kufareva, Irina

Ligand-Dependent Mechanisms of CC Chemokine Receptor 5 (CCR5) Trafficking Revealed by APEX2 Proximity Labeling Proteomics

APEX2邻近标记蛋白质组学揭示CC趋化因子受体5 (CCR5)转运的配体依赖性机制

Gu, Siyi; Maurya, Svetlana; Lona, Alexis; Borrega-Roman, Leire; Salanga, Catherina; Gonzalez, David J; Kufareva, Irina; Handel, Tracy M