日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Evaluation of a Boron-Conjugated SRC Inhibitor Combined with Proton and X-Ray Irradiation in U-87 MG and U-87 MG IDH1(R132H) Glioma Cell Lines.

对硼共轭 SRC 抑制剂与质子和 X 射线照射联合治疗 U-87 MG 和 U-87 MG IDH1(R132H) 胶质瘤细胞系的效果进行评价。

Alberghina Cristiana, Torrisi Filippo, Valable Samuel, Sarrazin Elsa, Blanchard Isis, Vela Anthony, Bravatà Valentina, Botta Lorenzo, Lanzanò Luca, Scalisi Silvia, Demichelis Maria P, Sabini Maria G, Patti Iolanda V, Russo Giorgio, Cammarata Francesco P, Parenti Rosalba

Modulation of the Antimelanoma Activity Imparted to Artemisinin Hybrids by the Monoterpene Counterpart

单萜类化合物对青蒿素杂合物抗黑色素瘤活性的调节

De Marchi, Elisa; Filippi, Silvia; Cesarini, Silvia; Di Maio, Beatrice; Bizzarri, Bruno Mattia; Saladino, Raffaele; Botta, Lorenzo

Serendipitous Identification of Azine Anticancer Agents Using a Privileged Scaffold Morphing Strategy.

利用优势骨架变形策略意外发现嗪类抗癌药物

Cesarini Silvia, Vicenti Ilaria, Poggialini Federica, Filippi Silvia, Mancin Eleonora, Fiaschi Lia, De Marchi Elisa, Giammarino Federica, Vagaggini Chiara, Bizzarri Bruno Mattia, Saladino Raffaele, Dreassi Elena, Zazzi Maurizio, Botta Lorenzo

Multicomponent Synthesis of C(8)-Substituted Purine Building Blocks of Peptide Nucleic Acids from Prebiotic Compounds

利用益生元化合物进行肽核酸C(8)取代嘌呤结构单元的多组分合成

Mancin, Eleonora; Capecchi, Eliana; Botta, Lorenzo; Bizzarri, Bruno Mattia

Molecular Dynamics Investigations of Human DNA-Topoisomerase I Interacting with Novel Dewar Valence Photo-Adducts: Insights into Inhibitory Activity

利用分子动力学方法研究人DNA拓扑异构酶I与新型杜瓦价光加合物的相互作用:对抑制活性的深入理解

Di Martino, Jessica; Arcieri, Manuel; Madeddu, Francesco; Pieroni, Michele; Carotenuto, Giovanni; Bottoni, Paolo; Botta, Lorenzo; Castrignanò, Tiziana; Gabellone, Sofia; Saladino, Raffaele

Synthesis of Artesunic Acid-Coumarin Hybrids as Potential Antimelanoma Agents

合成青蒿琥酯-香豆素杂合物作为潜在的抗黑色素瘤药物

Zippilli, Claudio; Filippi, Silvia; Cesarini, Silvia; Bizzarri, Bruno Mattia; Conigliaro, Pauline; De Marchi, Elisa; Botta, Lorenzo; Saladino, Raffaele

Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors

发现和优化新型大环脒基脲系列化合物,该系列化合物可作为酸性哺乳动物几丁质酶抑制剂

Balestri, Lorenzo Jacopo Ilic; Trivisani, Claudia Immacolata; Orofino, Francesco; Fiorucci, Diego; Truglio, Giuseppina Ivana; D'Agostino, Ilaria; Poggialini, Federica; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena

A Green Blue LED-Driven Two-Liquid-Phase One-Pot Procedure for the Synthesis of Estrogen-Related Quinol Prodrugs

一种绿蓝LED驱动的双液相一锅法合成雌激素相关醌类前药

De Marchi, Elisa; Botta, Lorenzo; Bizzarri, Bruno Mattia; Saladino, Raffaele

Investigation of fungal biomolecules after Low Earth Orbit exposure: a testbed for the next Moon missions

近地轨道暴露后真菌生物分子的研究:为下一次登月任务提供试验平台

Cassaro, Alessia; Pacelli, Claudia; Baqué, Mickael; Cavalazzi, Barbara; Gasparotto, Giorgio; Saladino, Raffaele; Botta, Lorenzo; Böttger, Ute; Rabbow, Elke; de Vera, Jean-Pierre; Onofri, Silvano

A Photochemoenzymatic Hunsdiecker-Borodin-Type Halodecarboxylation of Ferulic Acid

阿魏酸的光化学酶法Hunsdiecker-Borodin型卤代脱羧反应

Zippilli, Claudio; Bartolome, Miguel Jimenez; Hilberath, Thomas; Botta, Lorenzo; Hollmann, Frank; Saladino, Raffaele