日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Low-Efficacy Mu Opioid Agonists as Candidate Analgesics: Effects of Novel C-9 Substituted Phenylmorphans on Pain-Depressed Behavior in Mice.

低效μ阿片受体激动剂作为候选镇痛药:新型C-9取代苯基吗啡烷对小鼠疼痛抑制行为的影响

Santos Edna J, Akbarali Hamid I, Bow Eric W, Chambers Dana R, Gutman Eugene S, Jacobson Arthur E, Kang Minho, Lee Young K, Lutz Joshua A, Rice Kenner C, Sulima Agnieszka, Negus S Stevens

Discovery of a Potent Highly Biased MOR Partial Agonist among Diastereomeric C9-Hydroxyalkyl-5-phenylmorphans

在非对映异构体 C9-羟烷基-5-苯基吗啡烷中发现一种强效高偏向性 MOR 部分激动剂

Lutz, Joshua A; Sulima, Agnieszka; Gutman, Eugene S; Bow, Eric W; Luo, Dan; Kaska, Sophia; Prisinzano, Thomas E; Paronis, Carol A; Bergman, Jack; Imler, Gregory H; Kerr, Andrew T; Jacobson, Arthur E; Rice, Kenner C

Bivalent Conjugate Vaccine Induces Dual Immunogenic Response That Attenuates Heroin and Fentanyl Effects in Mice

二价结合疫苗诱导双重免疫反应,可减轻小鼠体内海洛因和芬太尼的作用

Barrientos, Rodell C; Whalen, Connor; Torres, Oscar B; Sulima, Agnieszka; Bow, Eric W; Komla, Essie; Beck, Zoltan; Jacobson, Arthur E; Rice, Kenner C; Matyas, Gary R

Novel Vaccine That Blunts Fentanyl Effects and Sequesters Ultrapotent Fentanyl Analogues

一种新型疫苗可减轻芬太尼的作用并隔离超强效芬太尼类似物

Barrientos, Rodell C; Bow, Eric W; Whalen, Connor; Torres, Oscar B; Sulima, Agnieszka; Beck, Zoltan; Jacobson, Arthur E; Rice, Kenner C; Matyas, Gary R