A small-molecule inverse agonist of PPARγ for advanced solid tumors: a phase 1 trial
用于治疗晚期实体瘤的小分子PPARγ反向激动剂:一项I期临床试验
期刊:Nature Medicine
影响因子:50
doi:10.1038/s41591-026-04263-3
Galsky, Matthew D; Mantia, Charlene; Bowden, Michaela; Bellmunt, Joaquim; Garmezy, Benjamin; Iyer, Gopa; Petrylak, Daniel P; Rasco, Drew; Gupta, Shilpa; Rodriguez-Rivera, Ildefonso; Mikhailov, Yelena; Joshi, Adarsh; Nguyen, Phuong A; Kakrecha, Bijal; Tepper, Jennifer; Costa, Anne Marie; McCrone, Carolyn; Rossi, Alex P; Mertz, Jennifer A; Gjini, Evisa; Meyers, Michael L; Milowsky, Matthew I; Gao, Xin