日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A high dose KRP203 induces cytoplasmic vacuoles associated with altered phosphoinositide segregation and endosome expansion

高剂量KRP203诱导细胞质空泡形成,并伴有磷脂酰肌醇分离异常和内体扩张。

Kofuji, Satoshi; Wolfe, Kara; Sumita, Kazutaka; Kageyama, Shun; Yoshino, Hirofumi; Hirota, Yoshihisa; Ogawa-Iio, Aki; Kanoh, Hirotaka; Sasaki, Mika; Kofuji, Kaori; Davis, Mindy I; Pragani, Rajan; Shen, Min; Boxer, Matthew B; Nakatsu, Fubito; Nigorikawa, Kiyomi; Sasaki, Takehiko; Takeuchi, Koh; Senda, Toshiya; Kim, Seong M; Edinger, Aimee L; Simeonov, Anton; Sasaki, Atsuo T

Multimodal action of KRP203 on phosphoinositide kinases in vitro and in cells

KRP203 在体外和细胞内对磷脂酰肌醇激酶的多模式作用

Ikeda, Yoshiki; Davis, Mindy I; Sumita, Kazutaka; Zheng, Yuxiang; Kofuji, Satoshi; Sasaki, Mika; Hirota, Yoshihisa; Pragani, Rajan; Shen, Min; Boxer, Matthew B; Takeuchi, Koh; Senda, Toshiya; Simeonov, Anton; Sasaki, Atsuo T

Discovery of novel inhibitors of human galactokinase by virtual screening

通过虚拟筛选发现人半乳糖激酶的新型抑制剂

Hu, Xin; Zhang, Ya-Qin; Lee, Olivia W; Liu, Li; Tang, Manshu; Lai, Kent; Boxer, Matthew B; Hall, Matthew D; Shen, Min

Canvass: A Crowd-Sourced, Natural-Product Screening Library for Exploring Biological Space

Canvass:一个用于探索生物空间的众包天然产物筛选库

Kearney, Sara E; Zahoránszky-Kőhalmi, Gergely; Brimacombe, Kyle R; Henderson, Mark J; Lynch, Caitlin; Zhao, Tongan; Wan, Kanny K; Itkin, Zina; Dillon, Christopher; Shen, Min; Cheff, Dorian M; Lee, Tobie D; Bougie, Danielle; Cheng, Ken; Coussens, Nathan P; Dorjsuren, Dorjbal; Eastman, Richard T; Huang, Ruili; Iannotti, Michael J; Karavadhi, Surendra; Klumpp-Thomas, Carleen; Roth, Jacob S; Sakamuru, Srilatha; Sun, Wei; Titus, Steven A; Yasgar, Adam; Zhang, Ya-Qin; Zhao, Jinghua; Andrade, Rodrigo B; Brown, M Kevin; Burns, Noah Z; Cha, Jin K; Mevers, Emily E; Clardy, Jon; Clement, Jason A; Crooks, Peter A; Cuny, Gregory D; Ganor, Jake; Moreno, Jesus; Morrill, Lucas A; Picazo, Elias; Susick, Robert B; Garg, Neil K; Goess, Brian C; Grossman, Robert B; Hughes, Chambers C; Johnston, Jeffrey N; Joullie, Madeleine M; Kinghorn, A Douglas; Kingston, David G I; Krische, Michael J; Kwon, Ohyun; Maimone, Thomas J; Majumdar, Susruta; Maloney, Katherine N; Mohamed, Enas; Murphy, Brian T; Nagorny, Pavel; Olson, David E; Overman, Larry E; Brown, Lauren E; Snyder, John K; Porco, John A Jr; Rivas, Fatima; Ross, Samir A; Sarpong, Richmond; Sharma, Indrajeet; Shaw, Jared T; Xu, Zhengren; Shen, Ben; Shi, Wei; Stephenson, Corey R J; Verano, Alyssa L; Tan, Derek S; Tang, Yi; Taylor, Richard E; Thomson, Regan J; Vosburg, David A; Wu, Jimmy; Wuest, William M; Zakarian, Armen; Zhang, Yufeng; Ren, Tianjing; Zuo, Zhong; Inglese, James; Michael, Sam; Simeonov, Anton; Zheng, Wei; Shinn, Paul; Jadhav, Ajit; Boxer, Matthew B; Hall, Matthew D; Xia, Menghang; Guha, Rajarshi; Rohde, Jason M

A Comprehensive Patient-Derived Xenograft Collection Representing the Heterogeneity of Melanoma

代表黑色素瘤异质性的综合性患者来源异种移植模型库

Krepler, Clemens; Sproesser, Katrin; Brafford, Patricia; Beqiri, Marilda; Garman, Bradley; Xiao, Min; Shannan, Batool; Watters, Andrea; Perego, Michela; Zhang, Gao; Vultur, Adina; Yin, Xiangfan; Liu, Qin; Anastopoulos, Ioannis N; Wubbenhorst, Bradley; Wilson, Melissa A; Xu, Wei; Karakousis, Giorgos; Feldman, Michael; Xu, Xiaowei; Amaravadi, Ravi; Gangadhar, Tara C; Elder, David E; Haydu, Lauren E; Wargo, Jennifer A; Davies, Michael A; Lu, Yiling; Mills, Gordon B; Frederick, Dennie T; Barzily-Rokni, Michal; Flaherty, Keith T; Hoon, Dave S; Guarino, Michael; Bennett, Joseph J; Ryan, Randall W; Petrelli, Nicholas J; Shields, Carol L; Terai, Mizue; Sato, Takami; Aplin, Andrew E; Roesch, Alexander; Darr, David; Angus, Steve; Kumar, Rakesh; Halilovic, Ensar; Caponigro, Giordano; Jeay, Sebastien; Wuerthner, Jens; Walter, Annette; Ocker, Matthias; Boxer, Matthew B; Schuchter, Lynn; Nathanson, Katherine L; Herlyn, Meenhard

PKM2 activation sensitizes cancer cells to growth inhibition by 2-deoxy-D-glucose

PKM2激活使癌细胞对2-脱氧-D-葡萄糖的生长抑制作用更加敏感

Tee, Sui Seng; Park, Jae Mo; Hurd, Ralph E; Brimacombe, Kyle R; Boxer, Matthew B; Massoud, Tarik F; Rutt, Brian K; Spielman, Daniel M

Corrigendum: A PHGDH inhibitor reveals coordination of serine synthesis and one-carbon unit fate

更正:PHGDH 抑制剂揭示了丝氨酸合成与一碳单元命运的协调性

Pacold, Michael E; Brimacombe, Kyle R; Chan, Sze Ham; Rohde, Jason M; Lewis, Caroline A; Swier, Lotteke J Y M; Possemato, Richard; Chen, Walter W; Sullivan, Lucas B; Fiske, Brian P; Cho, Steve; Freinkman, Elizaveta; Birsoy, Kıvanç; Abu, Monther-Remaileh; Shaul, Yoav D; Liu, Chieh Min; Zhou, Minerva; Koh, Min Jung; Chung, Haeyoon; Davidson, Shawn M; Luengo, Alba; Wang, Amy Q; Xu, Xin; Yasgar, Adam; Liu, Li; Rai, Ganesha; Westover, Kenneth D; Heiden, Matthew G Vander; Shen, Min; Gray, Nathanael S; Boxer, Matthew B; Sabatini, David M

Caspase-1 causes truncation and aggregation of the Parkinson's disease-associated protein α-synuclein

Caspase-1 会导致帕金森病相关蛋白 α-突触核蛋白的截断和聚集。

Wang, Wei; Nguyen, Linh T T; Burlak, Christopher; Chegini, Fariba; Guo, Feng; Chataway, Tim; Ju, Shulin; Fisher, Oriana S; Miller, David W; Datta, Debajyoti; Wu, Fang; Wu, Chun-Xiang; Landeru, Anuradha; Wells, James A; Cookson, Mark R; Boxer, Matthew B; Thomas, Craig J; Gai, Wei Ping; Ringe, Dagmar; Petsko, Gregory A; Hoang, Quyen Q

Identification of Novel Plasmodium falciparum Hexokinase Inhibitors with Antiparasitic Activity

鉴定具有抗寄生虫活性的新型恶性疟原虫己糖激酶抑制剂

Davis, Mindy I; Patrick, Stephen L; Blanding, Walker M; Dwivedi, Varun; Suryadi, Jimmy; Golden, Jennifer E; Coussens, Nathan P; Lee, Olivia W; Shen, Min; Boxer, Matthew B; Hall, Matthew D; Sharlow, Elizabeth R; Drew, Mark E; Morris, James C

PEPCK Coordinates the Regulation of Central Carbon Metabolism to Promote Cancer Cell Growth

PEPCK 协调中心碳代谢的调控以促进癌细胞生长

Montal, Emily D; Dewi, Ruby; Bhalla, Kavita; Ou, Lihui; Hwang, Bor Jang; Ropell, Ashley E; Gordon, Chris; Liu, Wan-Ju; DeBerardinis, Ralph J; Sudderth, Jessica; Twaddel, William; Boros, Laszlo G; Shroyer, Kenneth R; Duraisamy, Sekhar; Drapkin, Ronny; Powers, R Scott; Rohde, Jason M; Boxer, Matthew B; Wong, Kwok-Kin; Girnun, Geoffrey D