日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Alternative Approach to Sequence-Specific Recognition of DNA: Cooperative Stacking of Dication Dimers─Sensitivity to Compound Curvature, Aromatic Structure, and DNA Sequence

DNA序列特异性识别的替代方法:双阳离子二聚体的协同堆积——对化合物曲率、芳香结构和DNA序列的敏感性

Paul, Ananya; Terrell, J Ross; Farahat, Abdelbasset A; Ogbonna, Edwin N; Kumar, Arvind; Boykin, David W; Neidle, Stephen; Wilson, W David

Single GC base pair recognition by a heterocyclic diamidine: structures, affinities, and dynamics

杂环二脒对单个GC碱基对的识别:结构、亲和力和动力学

Ogbonna, Edwin N; Terrell, J Ross; Paul, Ananya; Farahat, Abdelbasset A; Poon, Gregory M K; Boykin, David W; Wilson, W David

Investigation of the effect of structure modification of furamidine on the DNA minor groove binding and antiprotozoal activity

研究呋喃脒结构修饰对DNA小沟结合及抗原生动物活性的影响

Farahat, Abdelbasset A; Kumar, Arvind; Wenzler, Tanja; Brun, Reto; Paul, Ananya; Guo, Pu; Wilson, W David; Boykin, David W

X-ray Structure Characterization of the Selective Recognition of AT Base Pair Sequences

AT碱基对序列选择性识别的X射线结构表征

Ogbonna, Edwin N; Paul, Ananya; Farahat, Abdelbasset A; Terrell, J Ross; Mineva, Ekaterina; Ogbonna, Victor; Boykin, David W; Wilson, W David

Arylimidamides Have Potential for Chemoprophylaxis against Blood-Transmitted Chagas Disease

芳基亚胺类药物具有预防血液传播的恰加斯病的潜力

Timm, Bruno Lisboa; da Gama, Aline Nefertiti Silva; Batista, Marcos Meuser; Batista, Denise da Gama Jaén; Boykin, David W; De Koning, Harry P; Correia Soeiro, Maria de Nazaré

Thermodynamic Factors That Drive Sequence-Specific DNA Binding of Designed, Synthetic Minor Groove Binding Agents

驱动设计合成的小沟结合剂与DNA序列特异性结合的热力学因素

Paul, Ananya; Farahat, Abdelbasset A; Boykin, David W; Wilson, W David

Dissecting Dynamic and Hydration Contributions to Sequence-Dependent DNA Minor Groove Recognition

剖析动态和水合作用对序列依赖性DNA小沟识别的影响

Ha, Van L T; Erlitzki, Noa; Farahat, Abdelbasset A; Kumar, Arvind; Boykin, David W; Poon, Gregory M K

A New Generation of Minor-Groove-Binding-Heterocyclic Diamidines That Recognize G·C Base Pairs in an AT Sequence Context

新一代识别AT序列中G·C碱基对的小沟结合杂环二脒类化合物

Paul, Ananya; Guo, Pu; Boykin, David W; Wilson, W David

Antileishmanial Efficacy and Pharmacokinetics of DB766-Azole Combinations

DB766-唑类药物组合的抗利什曼原虫疗效和药代动力学

Joice, April C; Yang, Sihyung; Farahat, Abdelbasset A; Meeds, Heidi; Feng, Mei; Li, Junan; Boykin, David W; Wang, Michael Zhuo; Werbovetz, Karl A

Phenotypic evaluation and in silico ADMET properties of novel arylimidamides in acute mouse models of Trypanosoma cruzi infection

在克氏锥虫感染急性小鼠模型中,对新型芳基酰胺类化合物进行表型评价和计算机模拟ADMET性质研究

da Silva, Cristiane França; Batista, Denise da Gama Jaén; de Araújo, Julianna Siciliano; Cunha-Junior, Edézio Ferreira; Stephens, Chad E; Banerjee, Moloy; Farahat, Abdelbasset A; Akay, Senol; Fisher, Mary K; Boykin, David W; Soeiro, Maria de Nazaré Correia