日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Genome-Guided Discovery of Antimalarial 4-Amino-2,4-Pentadienoate-Containing Cyclolipodepsipeptides

基因组引导的抗疟疾4-氨基-2,4-戊二烯酸酯环脂肽的发现

Candra, Hartono; Wang, Xue-Jiao; Go, Ka Diam; Feng, Li; Cai, Miaomiao; Ma, Guang-Lei; Widyantoro, Clarissa; Tan, Lik Tong; Bozdech, Zbynek; Wang, Zhe; Liang, Zhao-Xun

Mechanisms of PfDNMT2 inhibition and PfATP6-mediated resistance to the antimalarial candidate SC83288 in Plasmodium falciparum

恶性疟原虫中 PfDNMT2 抑制和 PfATP6 介导的抗疟候选药物 SC83288 耐药机制

Sanchez, Cecilia P; Duffey, Maëlle; Celada, Romina V; Kucharski, Michal; Hoarau, Marie; Saeyang, Thanaya; Kamchonwongpaisan, Sumalee; Sohraby, Farzin; de Buhr, Svenja; Nunes Alves, Ariane; Lucky, Amuza Byaruhanga; Miao, Jun; Regnault, Clement; Dziekan, Jerzy M; Bozdech, Zbynek; Barrett, Michael P; Lanzer, Michael

Integrative genomics of Plasmodium knowlesi reveals parasite-intrinsic regulators of severe human malaria

诺氏疟原虫的整合基因组学揭示了寄生虫自身控制严重人类疟疾的调控因子

Westaway, Jacob A F; Benavente, Ernest Diez; Kucharski, Michal; Nayak, Sourav; Huy, Duong T Q; Auburn, Sarah; William, Timothy; Rajahram, Giri S; Piera, Kim A; Trimarsanto, Hidayat; Hoon, Kian Soon; Bourke, Caitlin; Jantim, Anisah; Manah, Abdul Marsudi; Gotulis, William; Moon, Robert W; Amato, Roberto; Barber, Bridget E; Drakeley, Chris; Anstey, Nicholas M; Field, Matt A; Bozdech, Zbynek; Grigg, Matthew J

Plasmodiumfalciparum protein kinase 6 and hemozoin formation are inhibited by a type II human kinase inhibitor exhibiting antimalarial activity

一种具有抗疟活性的II型人激酶抑制剂可抑制恶性疟原虫蛋白激酶6和血红素的形成。

Flore Nardella ,Tiantian Jiang ,Lushun Wang ,Monica J Bohmer ,Subhoja Chakraborty ,John Okombo ,Jaeson Calla ,Tatiane Macedo Silva ,Samuel Pazicky ,Jianwei Che ,Jin Jeon ,Evie Vincent ,Nonlawat Boonyalai ,Rachael Coyle ,Mairi J Buchanan ,Samuel Schaefer ,Daisy Chen ,Amaan Khan ,Emily Mayville ,Mariana Laureano De Souza ,Mayland Treat ,Jordan Charlton ,Patrick K Tumwebaze ,Seth Tjia ,Lukas Montejo ,Karen Cover ,Philip J Rosenthal ,Roland A Cooper ,Zbynek Bozdech ,Marcus C S Lee ,Ratna Chakrabarti ,Sanjay A Desai ,David A Fidock ,Jinhua Wang ,Nathanael S Gray ,Elizabeth A Winzeler ,Debopam Chakrabarti

Characterizing the quick-killing mechanism of action of azithromycin analogs against malaria parasites

阐明阿奇霉素类似物对疟原虫的快速杀灭机制

Mao, Emma Y; Nguyen, William; Jana, Gouranga P; Maity, Bikash C; Pazicky, Samuel; Giannangelo, Carlo; Reader, Janette; Famodimu, Mufuliat T; Birkholtz, Lyn-Marie; Delves, Michael J; Creek, Darren J; Bozdech, Zbynek; Laleu, Benoît; Burrows, Jeremy N; Sleebs, Brad E; Gancheva, Maria R; Wilson, Danny W

Genomic epidemiology of Plasmodium knowlesi reveals putative genetic drivers of adaptation in Malaysia

诺氏疟原虫的基因组流行病学揭示了马来西亚适应性的潜在遗传驱动因素

Westaway, Jacob A F; Diez Benavente, Ernest; Auburn, Sarah; Kucharski, Michal; Aranciaga, Nicolas; Nayak, Sourav; William, Timothy; Rajahram, Giri S; Piera, Kim A; Braima, Kamil; Tan, Angelica F; Alaza, Danshy A; Barber, Bridget E; Drakeley, Chris; Amato, Roberto; Sutanto, Edwin; Trimarsanto, Hidayat; Jelip, Jenarun; Anstey, Nicholas M; Bozdech, Zbynek; Field, Matthew; Grigg, Matthew J

Identification of complex Plasmodium falciparum genetic backgrounds circulating in Africa: a multicountry genomic epidemiology analysis

非洲恶性疟原虫复杂遗传背景的鉴定:一项多国基因组流行病学分析

Miotto, Olivo; Amambua-Ngwa, Alfred; Amenga-Etego, Lucas N; Abdel Hamid, Muzamil M; Adam, Ishag; Aninagyei, Enoch; Apinjoh, Tobias; Awandare, Gordon A; Bejon, Philip; Bertin, Gwladys I; Bouyou-Akotet, Marielle; Claessens, Antoine; Conway, David J; D'Alessandro, Umberto; Diakite, Mahamadou; Djimdé, Abdoulaye; Dondorp, Arjen M; Duffy, Patrick; Fairhurst, Rick M; Fanello, Caterina I; Ghansah, Anita; Ishengoma, Deus S; Lawniczak, Mara; Maïga-Ascofaré, Oumou; Auburn, Sarah; Rosanas-Urgell, Anna; Wasakul, Varanya; White, Nina F D; Harrott, Alexandria; Almagro-Garcia, Jacob; Pearson, Richard D; Goncalves, Sonia; Ariani, Cristina; Bozdech, Zbynek; Hamilton, William L; Simpson, Victoria; Kwiatkowski, Dominic P

The artemisinin-induced dormant stages of Plasmodium falciparum exhibit hallmarks of cellular quiescence/senescence and drug resilience

青蒿素诱导的恶性疟原虫休眠期表现出细胞静止/衰老和耐药性的典型特征。

Tripathi, Jaishree; Stoklasa, Michal; Nayak, Sourav; En Low, Kay; Qian Hui Lee, Erica; Duong Tien, Quang Huy; Rénia, Laurent; Malleret, Benoit; Bozdech, Zbynek

Author Correction: The artemisinin-induced dormant stages of Plasmodium falciparum exhibit hallmarks of cellular quiescence/senescence and drug resilience

作者更正:青蒿素诱导的恶性疟原虫休眠期表现出细胞静止/衰老和耐药性的特征。

Tripathi, Jaishree; Stoklasa, Michal; Nayak, Sourav; En Low, Kay; Qian Hui Lee, Erica; Duong Tien, Quang Huy; Rénia, Laurent; Malleret, Benoit; Bozdech, Zbynek

Inhibition of falcilysin from Plasmodium falciparum by interference with its closed-to-open dynamic transition

通过干扰恶性疟原虫溶素的闭合-开放动态转变来抑制其活性

Lin, Jianqing; Yan, Xinfu; Chung, Zara; Liew, Chong Wai; El Sahili, Abbas; Pechnikova, Evgeniya V; Preiser, Peter R; Bozdech, Zbynek; Gao, Yong-Gui; Lescar, Julien