日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Potent Neuronal Nicotinamide Adenine Dinucleotide-Boosting Tetrahydroquinoxalines: Structure-Activity Relationships and Early Drug Metabolism and Pharmacokinetics Evaluation

强效神经元烟酰胺腺嘌呤二核苷酸增强型四氢喹喔啉类化合物:结构-活性关系及早期药物代谢和药代动力学评价

Cuřínová, Petra; Jöe, Melissa; Cesar, Filip; Nicol, Alan; Schwan, Kristián; Kohout, Michal; Varrichio, Carmine; Saleh, Aljona; Wheelock, Craig E; Jóhannesson, Gauti; Eigner, Václav; Tribble, James R; Brancale, Andrea; Williams, Pete A

Genome-wide meta-analysis identifies nine loci associated with higher risk of hepatocellular carcinoma development

全基因组荟萃分析确定了9个与肝细胞癌发生风险增加相关的基因位点。

Ghouse, Jonas; Gellert-Kristensen, Helene; O'Rourke, Colm J; Seidelin, Anne-Sofie; Thorleifsson, Gudmar; Sveinbjörnsson, Gardar; Tragante, Vinicius; Konkwo, Chigoziri; Brancale, Joseph; Vilarinho, Silvia; Eyrich, Tim M; Ahlberg, Gustav; Bundgaard, Johan S; Rand, Søren A; Lundegaard, Pia R; Sørensen, Erik; Mikkelsen, Christina; Træholt, Jacob; Erikstrup, Christian; Dinh, Khoa M; Bruun, Mie T; Jensen, Bitten Aa; Bay, Jakob T; Brunak, Søren; Banasik, Karina; Ullum, Henrik; Laisk, Triin; Mägi, Reedik; Nadauld, Lincoln D; Knowlton, Kirk U; Knight, Stacey; Gluud, Lise L; Vistisen, Kirsten; Björnsson, Einar S; Ulfarsson, Magnus O; Sulem, Patrick; Holm, Hilma; Pedersen, Ole B; Ostrowski, Sisse R; Gudbjartsson, Daniel F; Rafnar, Thorunn; Stefansson, Kari; Lassen, Ulrik; Pommergaard, Hans-Christian; Hillingsø, Jens G; Andersen, Jesper B; Bundgaard, Henning; Stender, Stefan

Correction: Impairment of cocaine-mediated behaviours in mice by clinically relevant Ras-ERK inhibitors

更正:临床相关Ras-ERK抑制剂对小鼠可卡因介导行为的损害

Papale, Alessandro; Morella, Ilaria Maria; Indrigo, Marzia Tina; Bernardi, Rick E; Marrone, Livia; Marchisella, Francesca; Brancale, Andrea; Spanagel, Rainer; Brambilla, Riccardo; Fasano, Stefania

Quinoxaline-based anti-schistosomal compounds have potent anti-plasmodial activity.

喹喔啉类抗血吸虫化合物具有很强的抗疟原虫活性

Rawat Mukul, Padalino Gilda, Adika Edem, Okombo John, Yeo Tomas, Brancale Andrea, Fidock David A, Hoffmann Karl F, Lee Marcus C S

New dengue virus inhibitors targeting NS3-NS5 interaction identified by in silico screening

通过计算机筛选发现靶向NS3-NS5相互作用的新型登革病毒抑制剂

Nannetti, Giulio; Mercorelli, Beatrice; Bazzacco, Alessandro; Santi, Nicolò; Celegato, Marta; Ferla, Salvatore; Sturlese, Mattia; Buurma, Niklaas J; Brancale, Andrea; Loregian, Arianna

Stereoanalysis of the Antiparasitic Natural Product Callunene and Its Synthetic Intermediates

抗寄生虫天然产物卡鲁烯及其合成中间体的立体分析

Ferenczei, Jiří; Blahout, Vilém; Dvořáková, Hana; Brancale, Andrea; Cuřínová, Petra; Labíková, Magdaléna; Kohout, Michal; Setnička, Vladimír; Perlíková, Pavla

New Anticancer 4-Aryldihydropyrimidinone-5-Carboxylates Targeting Hsp90.

靶向 Hsp90 的新型抗癌 4-芳基二氢嘧啶酮-5-羧酸酯。

Bordoni Cinzia, Elstow Tia Z, Brancale Andrea, Clarkson Richard W E, Westwell Andrew D

Substituent-Driven Anion-Binding Selectivity in Aliphatic Chain-Substituted 1,2-Phenylene Urea Macrocycles and Optimized Synthetic Methodology

脂肪链取代的1,2-亚苯基脲大环化合物中取代基驱动的阴离子结合选择性及优化的合成方法

Svobodová, Kateřina; Eigner, Václav; Brancale, Andrea; Cuřínová, Petra; Himl, Michal

Germline Variants Influence Chronic Liver Disease Progression through Distinct Pathways

种系变异通过不同的途径影响慢性肝病进展

Vujkovic, Marijana; Kaplan, David E; Ghouse, Jonas; Loza, Bao-Li; Brancale, Joseph; Lewis, Adam; Zhang, David Y; Levin, Michael G; Veatch, Olivia J; Johnson, Josephine P; Schneider, Carolin V; Verma, Anurag; Wangensteen, Kirk J; Scorletti, Eleonora; Gill, Dipender; Konkwo, Chigoziri; Garófalo, Alexis M; Guare, Lindsay A; Schwantes-An, Tae-Wi; Abreu, Marco V; Gellert-Kristensen, Helene; Pedersen, Ole B; Erikstrup, Christian; Bundgaard, Johan S; Sørensen, Erik; Ostrowski, Sisse R; Bundgaard, Henning; Lee, Kyung Min; Shaked, Abraham; Olthoff, Kim M; Hoteit, Maarouf A; Speliotes, Elizabeth K; Chen, Yanhua; Oliveri, Antonino; Yin, Lishi; Valenti, Luca Vc; Malvestiti, Francesco; Marchelli, Daniele; Miano, Lorenzo; Anstee, Quentin M; Daly, Ann K; Cordell, Heather J; Darlay, Rebecca; Verweij, Niek; Hindy, George; Locke, Adam; Matsuura, Kentaro; Asrani, Sumeet K; Testa, Giuliano; Lotta, Luca A; Jones, Marcus B; Dochtermann, Daniel R; Norden-Krichmar, Trina M; Teerlink, Craig C; Devineni, Poornima; Pyarajan, Saiju; Rader, Daniel J; Tanaka, Yasuhito; Voight, Benjamin F; Vilarinho, Silvia; Bastarache, Lisa A; Stender, Stefan; Tsao, Philip S; Morgan, Timothy R; Lynch, Julie A; Chang, Kyong-Mi

Multifaceted roles for BCL3 in cancer: a proto-oncogene comes of age

BCL3在癌症中的多重作用:一种原癌基因走向成熟

Seaton, Gillian; Smith, Hannah; Brancale, Andrea; Westwell, Andrew D; Clarkson, Richard