日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

In vitro toxicokinetics and metabolic profiling of methoxycathinones and methylthiocathinones using human liver systems and hyphenated mass spectrometry

利用人肝系统和联用质谱法对甲氧基卡西酮和甲基硫代卡西酮进行体外毒代动力学和代谢分析

期刊:Archives of Toxicology
影响因子:6.9
doi:10.1007/s00204-025-04205-x
Kroesen, Matthias D; Gampfer, Tanja M; Wagmann, Lea; Kavanagh, Pierce V; Brandt, Simon D; Meyer, Markus R
代谢
发表日期：2026
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Bioisostere-Driven Discovery of SePP: A Selenium-Containing Polypharmacological Agent Relevant to Fragile X Syndrome

生物等排体驱动的SePP发现：一种与脆性X综合征相关的含硒多药理学药物

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c02700
Wallach, Jason; Cameron, Sean; Dybek, Michael; Stanley, Branden; Orme, Christopher; Riad, Nour; Kavanagh, Pierce; Brandt, Simon D; Knapp, Adam; Gamrat, James; Jauhola-Straight, Rebekah; Adejare, Adeboye; Rogier, Alexander J; Tyagi, Richa; Canal, Clinton E
发表日期：2026
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Prolintane analogs as hybrid monoamine transporter ligands: Structural determinants and species differences

脯氨酰胺类似物作为杂合单胺转运体配体：结构决定因素和物种差异

期刊:Journal of Biological Chemistry
影响因子:3.9
doi:10.1016/j.jbc.2025.110903
Kastner, Nina; Islam, Mohammad N; Dybek, Michael; Roth, Evelyn; Heisinger, Simon; Holy, Marion; Jäntsch, Kathrin; Walther, Donna; Stockner, Thomas; Baumann, Michael H; Brandt, Simon D; Wallach, Jason; Sitte, Harald H; Kudlacek, Oliver
发表日期：2025
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A Comparative Study Using Reversed-Phase and Hydrophilic Interaction Liquid Chromatography to Investigate the In Vitro and In Vivo Metabolism of Five Selenium-Containing Cathinone Derivatives

采用反相和亲水相互作用液相色谱法对五种含硒卡西酮衍生物的体外和体内代谢进行比较研究

期刊:Metabolites
影响因子:3.7
doi:10.3390/metabo15080497
Wagmann, Lea; Schmitt, Jana H; Gampfer, Tanja M; Brandt, Simon D; Scott, Kenneth; Kavanagh, Pierce V; Meyer, Markus R
代谢
发表日期：2025
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Bioisosteric analogs of MDMA: Improving the pharmacological profile?

MDMA的生物等排体类似物：能否改善其药理特性？

期刊:Journal of Neurochemistry
影响因子:4
doi:10.1111/jnc.16149
Alberto-Silva Ana Sofia, Hemmer Selina, Bock Hailey A, da Silva Leticia Alves, Scott Kenneth R, Kastner Nina, Bhatt Manan, Niello Marco, Jäntsch Kathrin, Kudlacek Oliver, Bossi Elena, Stockner Thomas, Meyer Markus R, McCorvy John D, Brandt Simon D, Kavanagh Pierce, Sitte Harald H
其它
发表日期：2024
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Bioisosteric analogs of MDMA with improved pharmacological profile

具有改进药理特性的MDMA生物等排体类似物

期刊:
影响因子:
doi:10.1101/2024.04.08.588083
Alberto-Silva, Ana Sofia; Hemmer, Selina; Bock, Hailey A; Alves da Silva, Leticia; Scott, Kenneth R; Kastner, Nina; Bhatt, Manan; Niello, Marco; Jäntsch, Kathrin; Kudlacek, Oliver; Bossi, Elena; Stockner, Thomas; Meyer, Markus R; McCorvy, John D; Brandt, Simon D; Kavanagh, Pierce; Sitte, Harald H
发表日期：2024
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Use of the head-twitch response to investigate the structure-activity relationships of 4-thio-substituted 2,5-dimethoxyphenylalkylamines

利用头部抽搐反应研究4-硫代取代的2,5-二甲氧基苯基烷基胺的构效关系

期刊:Psychopharmacology
影响因子:3.3
doi:10.1007/s00213-022-06279-2
Halberstadt, Adam L; Luethi, Dino; Hoener, Marius C; Trachsel, Daniel; Brandt, Simon D; Liechti, Matthias E
发表日期：2023
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(2-Aminopropyl)benzo[β]thiophenes (APBTs) are novel monoamine transporter ligands that lack stimulant effects but display psychedelic-like activity in mice

(2-氨丙基)苯并[β]噻吩 (APBTs) 是一类新型单胺转运体配体，它们不具有兴奋作用，但在小鼠体内却表现出类似迷幻剂的活性。

期刊:Neuropsychopharmacology
影响因子:7.1
doi:10.1038/s41386-021-01221-0
Rudin, Deborah; McCorvy, John D; Glatfelter, Grant C; Luethi, Dino; Szöllősi, Dániel; Ljubišić, Tea; Kavanagh, Pierce V; Dowling, Geraldine; Holy, Marion; Jaentsch, Kathrin; Walther, Donna; Brandt, Simon D; Stockner, Thomas; Baumann, Michael H; Halberstadt, Adam L; Sitte, Harald H
发表日期：2022
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Investigation of the Structure-Activity Relationships of Psilocybin Analogues

裸盖菇素类似物结构-活性关系的研究

期刊:ACS Pharmacology and Translational Science
影响因子:3.7
doi:10.1021/acsptsci.0c00176
Klein, Adam K; Chatha, Muhammad; Laskowski, Lauren J; Anderson, Emilie I; Brandt, Simon D; Chapman, Stephen J; McCorvy, John D; Halberstadt, Adam L
发表日期：2021
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Pharmacological and biotransformation studies of 1-acyl-substituted derivatives of d-lysergic acid diethylamide (LSD)

d-麦角酸二乙酰胺（LSD）1-酰基取代衍生物的药理学和生物转化研究

期刊:Neuropharmacology
影响因子:4.6
doi:10.1016/j.neuropharm.2019.107856
Halberstadt, Adam L; Chatha, Muhammad; Klein, Adam K; McCorvy, John D; Meyer, Markus R; Wagmann, Lea; Stratford, Alexander; Brandt, Simon D
发表日期：2020
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