日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: Tumor Microenvironment Landscapes Supporting EGFR-mutant NSCLC Are Modulated at the Single-cell Interaction Level by Unesbulin Treatment

更正:Unesbulin治疗在单细胞相互作用水平上调节支持EGFR突变型非小细胞肺癌的肿瘤微环境图谱

Maroni, Giorgia; Krishnan, Indira; Alfieri, Roberta; Maymi, Valerie A; Pandell, Nicole; Csizmadia, Eva; Zhang, Junyan; Weetall, Marla; Branstrom, Art; Braccini, Giulia; San Millán, Eva Cabrera; Storti, Barbara; Bizzarri, Ranieri; Kocher, Olivier; Bassères, Daniela S; Welner, Robert S; Magli, Maria Cristina; Merelli, Ivan; Clohessy, John G; Ali, Azhar; Tenen, Daniel G; Levantini, Elena

Tumor Microenvironment Landscapes Supporting EGFR-mutant NSCLC Are Modulated at the Single-cell Interaction Level by Unesbulin Treatment

Unesbulin治疗在单细胞相互作用水平上调节支持EGFR突变型非小细胞肺癌的肿瘤微环境图谱

Giorgia Maroni ,Indira Krishnan # ,Roberta Alfieri # ,Valerie A Maymi ,Nicole Pandell ,Eva Csizmadia ,Junyan Zhang ,Marla Weetall ,Art Branstrom ,Giulia Braccini ,Eva Cabrera San Millán ,Barbara Storti ,Ranieri Bizzarri ,Olivier Kocher ,Daniela S Daniela Sanchez Bassères ,Robert S Welner ,Maria Cristina Magli ,Ivan Merelli ,John G Clohessy ,Azhar Ali # ,Daniel G Tenen # ,Elena Levantini #

Emvododstat, a Potent Dihydroorotate Dehydrogenase Inhibitor, Is Effective in Preclinical Models of Acute Myeloid Leukemia

Emvododstat 是一种有效的二氢乳清酸脱氢酶抑制剂,对急性髓系白血病的临床前模型有效

Arthur Branstrom, Liangxian Cao, Bansri Furia, Christopher Trotta, Marianne Santaguida, Jason D Graci, Joseph M Colacino, Balmiki Ray, Wencheng Li, Josephine Sheedy, Anna Mollin, Shirley Yeh, Ronald Kong, Richard Sheridan, John D Baird, Kylie O'Keefe, Robert Spiegel, Elizabeth Goodwin, Suzanne Keati

Preclinical and Early Clinical Development of PTC596, a Novel Small-Molecule Tubulin-Binding Agent

新型小分子微管蛋白结合剂PTC596的临床前和早期临床开发

Jernigan, Finith; Branstrom, Arthur; Baird, John D; Cao, Liangxian; Dali, Mandar; Furia, Bansri; Kim, Min Jung; O'Keefe, Kylie; Kong, Ronald; Laskin, Oscar L; Colacino, Joseph M; Pykett, Mark; Mollin, Anna; Sheedy, Josephine; Dumble, Melissa; Moon, Young-Choon; Sheridan, Richard; Mühlethaler, Tobias; Spiegel, Robert J; Prota, Andrea E; Steinmetz, Michel O; Weetall, Marla

Effective Delivery of a Microtubule Polymerization Inhibitor Synergizes with Standard Regimens in Models of Pancreatic Ductal Adenocarcinoma

微管聚合抑制剂的有效递送与胰腺导管腺癌模型中的标准方案产生协同作用

Jaime A Eberle-Singh, Irina Sagalovskiy, H Carlo Maurer, Stephen A Sastra, Carmine F Palermo, Amanda R Decker, Min Jung Kim, Josephine Sheedy, Anna Mollin, Liangxian Cao, Jianhua Hu, Arthur Branstrom, Marla Weetall, Kenneth P Olive

Discovery and Optimization of Indolyl-Containing 4-Hydroxy-2-Pyridone Type II DNA Topoisomerase Inhibitors Active against Multidrug Resistant Gram-negative Bacteria

发现和优化含吲哚基的4-羟基-2-吡啶酮II型DNA拓扑异构酶抑制剂,该抑制剂对多重耐药革兰氏阴性菌具有活性

Gerasyuto, Aleksey I; Arnold, Michael A; Wang, Jiashi; Chen, Guangming; Zhang, Xiaoyan; Smith, Sean; Woll, Matthew G; Baird, John; Zhang, Nanjing; Almstead, Neil G; Narasimhan, Jana; Peddi, Srinivasa; Dumble, Melissa; Sheedy, Josephine; Weetall, Marla; Branstrom, Arthur A; Prasad, J V N; Karp, Gary M

Inhibition of BMI1, a Therapeutic Approach in Endometrial Cancer

抑制BMI1是子宫内膜癌的一种治疗方法

Megan Buechel # ,Anindya Dey # ,Shailendra Kumar Dhar Dwivedi ,Aleia Crim ,Kai Ding ,Roy Zhang ,Priyabrata Mukherjee ,Kathleen N Moore ,Liangxian Cao ,Arthur Branstrom ,Marla Weetall ,John Baird ,Resham Bhattacharya

The minor gentamicin complex component, X2, is a potent premature stop codon readthrough molecule with therapeutic potential

庆大霉素复合物的次要成分 X2 是一种有效的提前终止密码子读通分子,具有治疗潜力

Westley J Friesen, Briana Johnson, Jairo Sierra, Jin Zhuo, Priya Vazirani, Xiaojiao Xue, Yuki Tomizawa, Ramil Baiazitov, Christie Morrill, Hongyu Ren, Suresh Babu, Young-Choon Moon, Art Branstrom, Anna Mollin, Jean Hedrick, Josephine Sheedy, Gary Elfring, Marla Weetall, Joseph M Colacino, Ellen M We

Targeting of BMI-1 expression by the novel small molecule PTC596 in mantle cell lymphoma

新型小分子PTC596靶向套细胞淋巴瘤中的BMI-1表达

Maeda, Aya; Nishida, Yuki; Weetall, Marla; Cao, Liangxian; Branstrom, Arthur; Ishizawa, Jo; Nii, Takenobu; Schober, Wendy D; Abe, Yoshiaki; Matsue, Kosei; Yoshimura, Mariko; Kimura, Shinya; Kojima, Kensuke

The novel BMI-1 inhibitor PTC596 downregulates MCL-1 and induces p53-independent mitochondrial apoptosis in acute myeloid leukemia progenitor cells

新型 BMI-1 抑制剂 PTC596 可下调 MCL-1 并诱导急性髓系白血病祖细胞中 p53 独立的线粒体凋亡

Y Nishida, A Maeda, M J Kim, L Cao, Y Kubota, J Ishizawa, A AlRawi, Y Kato, A Iwama, M Fujisawa, K Matsue, M Weetall, M Dumble, M Andreeff, T W Davis, A Branstrom, S Kimura, K Kojima