Targeting the Main Protease (M(pro), nsp5) by Growth of Fragment Scaffolds Exploiting Structure-Based Methodologies
利用基于结构的方法,通过片段支架的生长来靶向主要蛋白酶(M(pro), nsp5)
期刊:ACS Chemical Biology
影响因子:3.8
doi:10.1021/acschembio.3c00720
Altincekic, Nadide; Jores, Nathalie; Löhr, Frank; Richter, Christian; Ehrhardt, Claus; Blommers, Marcel J J; Berg, Hannes; Öztürk, Sare; Gande, Santosh L; Linhard, Verena; Orts, Julien; Abi Saad, Marie Jose; Bütikofer, Matthias; Kaderli, Janina; Karlsson, B Göran; Brath, Ulrika; Hedenström, Mattias; Gröbner, Gerhard; Sauer, Uwe H; Perrakis, Anastassis; Langer, Julian; Banci, Lucia; Cantini, Francesca; Fragai, Marco; Grifagni, Deborah; Barthel, Tatjana; Wollenhaupt, Jan; Weiss, Manfred S; Robertson, Angus; Bax, Adriaan; Sreeramulu, Sridhar; Schwalbe, Harald