日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Utilizing Constrained Bicyclic Peptides for In Vitro Diagnostics.

利用受限双环肽进行体外诊断。

Shamsabadi André, Creamer Adam, Sadler Christy J, Abdelwahed Aida, Gaynor Katherine U, Demydchuk Yuliya, Ivanova-Berndt Gabriela, Van Rietschoten Katerine, Beswick Paul, Chen Liuhong, Arruda Bezerra Gustavo, Lulla Aleksei, Brear Paul, Hyvönen Marko, Skynner Michael J, Stevens Molly M

Yeast Display Technology Enables Rapid Discovery of Low-Nanomolar Macrocyclic Peptide Inhibitors of Human Angiotensin-Converting Enzyme 2

酵母展示技术可快速发现低纳摩尔级人血管紧张素转化酶2大环肽抑制剂

Romanyuk, Zhanna; Bettin, Giacomo; Brear, Paul; Linciano, Sara; Mazzocato, Ylenia; Bonadies, Simone; Zanotto, Ilaria; Mazzucco, Camilla; Monferone, Alan; Soler, Miguel A; Pasut, Gianfranco; Martin, Sara De; Scarso, Alessandro; Heinis, Christian; Rothenberger, Sylvia; Hyvönen, Marko; Angelini, Alessandro

Rapid discovery of monoclonal antibodies by microfluidics-enabled FACS of single pathogen-specific antibody-secreting cells

利用微流控技术对单个病原体特异性抗体分泌细胞进行流式细胞术分选,快速发现单克隆抗体

Katrin Fischer ,Aleksei Lulla # ,Tsz Y So # ,Pehuén Pereyra-Gerber # ,Matthew I J Raybould # ,Timo N Kohler # ,Juan Carlos Yam-Puc # ,Tomasz S Kaminski ,Robert Hughes ,Gwendolyn L Pyeatt ,Florian Leiss-Maier ,Paul Brear ,Nicholas J Matheson ,Charlotte M Deane ,Marko Hyvönen ,James E D Thaventhiran ,Florian Hollfelder

Potent Fluorescent Probe for Target-Engagement Studies of Allosteric Pyruvate Kinase Modulators

用于变构丙酮酸激酶调节剂靶点结合研究的高效荧光探针

Nilsson, Oscar; Valaka, Anna P; Håversen, Liliana; Bogucka, Agnieszka; Köteles, István; Brear, Paul; Rutberg, Mikael; Gunnarsson, Anders; Hyvönen, Marko; Grøtli, Morten

Transcriptome-scale analysis uncovers conserved residues in the hydrophobic core of the bacterial RNA chaperone Hfq required for small regulatory RNA stability

转录组规模分析揭示了细菌 RNA 伴侣 Hfq 疏水核心中保守的残基,这些残基是小调节 RNA 稳定性所必需的

Josh McQuail, Miroslav Krepl, Kai Katsuya-Gaviria, Aline Tabib-Salazar, Lynn Burchell, Thorsten Bischler, Tom Gräfenhan, Paul Brear, Jiří Šponer, Ben F Luisi, Sivaramesh Wigneshweraraj

Exploiting the Cryptic αD Pocket of Casein Kinase 2α (CK2α) to Deliver Highly Potent and Selective Type 1 Inhibitors.

利用酪蛋白激酶 2α (CK2α) 的隐蔽 αD 口袋递送高效选择性 1 型抑制剂。

Glossop Paul A, Brear Paul, Wright Susanne, Flanagan Neil, Glossop Melanie S, Lane Charlotte A L, Butt Richard P, Spring David R, Hyvönen Marko, Cawkill Darren

Investigation into the effect of phenylalanine gating on anaerobic haem breakdown using the energy landscape approach

利用能量景观方法研究苯丙氨酸门控对厌氧血红素分解的影响

Keith, Alasdair D; Sawyer, Elizabeth B; Choy, Desmond C Y; Cole, James L; Shang, Cheng; Biggs, George S; Klein, Oskar James; Brear, Paul D; Wales, David J; Barker, Paul D

Using electricity tariffs and thermal comfort management to promote residential energy decarbonization

利用电价和热舒适管理促进住宅能源脱碳

Vecchi, Andrea; Brear, Michael John

The 2-methylcitrate cycle and the glyoxylate shunt in Pseudomonas aeruginosa are linked through enzymatic redundancy

铜绿假单胞菌中的2-甲基柠檬酸循环和乙醛酸循环通过酶冗余联系在一起。

Wijaya, Andre J; Dolan, Stephen K; Kohlstedt, Michael; Gläser, Lars; Brear, Paul; Geddis, Stephen; Wittmann, Christoph; Spring, David R; Welch, Martin

Pseudomonas aeruginosa PfpI is a methylglyoxalase

铜绿假单胞菌 PfpI 是一种甲基乙二醛酶

Grimm, Larson; Wijaya, Andre; Askenasy, Isabel; Nazeer, Rahan Rudland; Seki, Hikaru; Brear, Paul D; Figueroa, Wendy; Spring, David R; Welch, Martin