日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

ReCHEMbinant stapling enhances intracellular delivery and bioactivity of engineered protein inhibitors

ReCHEMbinant 交联技术可增强工程化蛋白抑制剂的细胞内递送和生物活性。

Kahler, Jan Pascal; Ellenbroek, Brecht D; van der Noord, Vera E; van de Water, Bob; Pomplun, Sebastian J

Development of DuoMYC: a synthetic cell penetrant miniprotein that efficiently inhibits the oncogenic transcription factor MYC

DuoMYC的研发:一种能有效抑制致癌转录因子MYC的合成细胞穿透性小蛋白

Ellenbroek, Brecht D; Kahler, Jan Pascal; Arella, Damiano; Lin, Cherina; Jespers, Willem; Züger, Eliane Ann-Katrin; Drukker, Micha; Pomplun, Sebastian J

AlphaFold-Guided Discovery of an Overlapping MYC/Miz-1 Interface Enables Peptidomimetic Disruption of MYC/MAX

AlphaFold引导发现重叠的MYC/Miz-1界面,从而实现肽模拟物对MYC/MAX的破坏

Ellenbroek, Brecht D; Tirtosentono, Amardhiko S S; Pomplun, Sebastian J

Identification of an alternative triglyceride biosynthesis pathway

鉴定出一条替代的甘油三酯生物合成途径

Gian-Luca McLelland ,Marta Lopez-Osias ,Cristy R C Verzijl ,Brecht D Ellenbroek ,Rafaela A Oliveira ,Nicolaas J Boon ,Marleen Dekker ,Lisa G van den Hengel ,Rahmen Ali ,Hans Janssen ,Ji-Ying Song ,Paul Krimpenfort ,Tim van Zutphen ,Johan W Jonker ,Thijn R Brummelkamp

Stereoselective Synthesis of Fused Vinylcyclopropanes by Intramolecular Tsuji-Trost Cascade Cyclization

通过分子内辻-特罗斯特级联环化反应立体选择性合成稠合乙烯基环丙烷

Braun, John; Ariëns, Maxim I; Matsuo, Bianca T; de Vries, Steven; van Wordragen, Ellen D H; Ellenbroek, Brecht D; Vande Velde, Christophe M L; Orru, Romano V A; Ruijter, Eelco