日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of AZD4144, a Selective and Potent NLRP3 Inhibitor for the Treatment of Inflammatory Diseases.

发现 AZD4144,一种选择性强效的 NLRP3 抑制剂,可用于治疗炎症性疾病

Johansson Anders, Sugama Hiroshi, Larsson Niklas, Winiwarter Susanne, Yoshida Kosuke, Gradén Henrik, Bergonzini Giulia, Matsumura Takehiko, Miyazaki Shiki, Fuchigami Ryuichi, Eda Masahiro, Takamatsu Hisayuki, Iguchi Kaori, Hongu Mitsuya, Matsudaira Tetsuji, Hovdal Daniel, Fredenwall Marlene, Fahlander Ulf, Luchniak Anna, Brengdahl Johan, Jung Bomi, Rhedin Magdalena, Sardana Juhi, Idei Akiko, Kato Yosuke, Kimura Junpei, Viklund Jenny, Brandt Peter, Sjögren Anna-Karin, Hibino Yui, Woollard Kevin, Yoneda Hikaru

Design of Selective sPLA(2)-X Inhibitor (-)-2-{2-[Carbamoyl-6-(trifluoromethoxy)-1H-indol-1-yl]pyridine-2-yl}propanoic Acid

选择性 sPLA(2)-X 抑制剂 (-)-2-{2-[氨基甲酰基-6-(三氟甲氧基)-1H-吲哚-1-基]吡啶-2-基}丙酸的设计

Giordanetto, Fabrizio; Knerr, Laurent; Nordberg, Peter; Pettersen, Daniel; Selmi, Nidhal; Beisel, Hans-Georg; de la Motte, Hannah; Månsson, Åsa; Dahlström, Mikael; Broddefalk, Johan; Saarinen, Gabrielle; Klingegård, Fredrik; Hurt-Camejo, Eva; Rosengren, Birgitta; Wikström, Johannes; Wågberg, Maria; Brengdahl, Johan; Rohman, Mattias; Sandmark, Jenny; Åkerud, Tomas; Roth, Robert G; Jansen, Frank; Ahlqvist, Marie

Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A(2) Type X (sPLA(2)-X) Inhibitors.

发现一系列吲哚-2 甲酰胺类化合物作为选择性分泌型磷脂酶 A(2) X 型 (sPLA(2)-X) 抑制剂

Knerr Laurent, Giordanetto Fabrizio, Nordberg Peter, Pettersen Daniel, Selmi Nidhal, Beisel Hans-Georg, de la Motte Hannah, Olsson Thomas, Perkins Tim D J, Herslöf Margareta, Månsson à sa, Dahlström Mikael, Starke Ingemar, Broddefalk Johan, Saarinen Gabrielle, Klingegård Fredrik, Hurt-Camejo Eva, Rosengren Birgitta, Brengdahl Johan, Jansen Frank, Rohman Mattias, Sandmark Jenny, Hallberg Kenth, à kerud Tomas, Roth Robert G, Ahlqvist Marie

Novel Zn2+ Modulated GPR39 Receptor Agonists Do Not Drive Acute Insulin Secretion in Rodents

新型 Zn2+ 调节的 GPR39 受体激动剂不会诱导啮齿动物急性胰岛素分泌

Fjellström, Ola; Larsson, Niklas; Yasuda, Shin-Ichiro; Tsuchida, Takuma; Oguma, Takahiro; Marley, Anna; Wennberg-Huldt, Charlotte; Hovdal, Daniel; Fukuda, Hajime; Yoneyama, Yukimi; Sasaki, Kazuyo; Johansson, Anders; Lundqvist, Sara; Brengdahl, Johan; Isaacs, Richard J; Brown, Daniel; Geschwindner, Stefan; Benthem, Lambertus; Priest, Claire; Turnbull, Andrew