Discovery of CP-690,550: a potent and selective Janus kinase (JAK) inhibitor for the treatment of autoimmune diseases and organ transplant rejection
发现 CP-690,550:一种强效且选择性的 Janus 激酶 (JAK) 抑制剂,用于治疗自身免疫性疾病和器官移植排斥
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm1004286
Mark E Flanagan, Todd A Blumenkopf, William H Brissette, Matthew F Brown, Jeffrey M Casavant, Chang Shang-Poa, Jonathan L Doty, Eileen A Elliott, Michael B Fisher, Michael Hines, Craig Kent, Elizabeth M Kudlacz, Brett M Lillie, Kelly S Magnuson, Sandra P McCurdy, Michael J Munchhof, Bret D Perry, Pe