日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Niacin lipid efficacy is independent of both the niacin receptor GPR109A and free fatty acid suppression

烟酸脂质功效与烟酸受体 GPR109A 和游离脂肪酸抑制无关

Brett Lauring, Andrew K P Taggart, James R Tata, Richard Dunbar, Luzelena Caro, Kang Cheng, Jayne Chin, Steven L Colletti, Josee Cote, Sauzanne Khalilieh, Jiajun Liu, Wen-Lin Luo, Alexandra A Maclean, Laurence B Peterson, Adam B Polis, Waheeda Sirah, Tsuei-Ju Wu, Xuan Liu, Lan Jin, Kenneth Wu, P Dou

(1aR,5aR)1a,3,5,5a-Tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (MK-1903): a potent GPR109a agonist that lowers free fatty acids in humans

(1aR,5aR)1a,3,5,5a-四氢-1H-2,3-二氮杂-环丙基[a]戊二烯-4-羧酸 (MK-1903):一种有效的 GPR109a 激动剂,可降低人类体内的游离脂肪酸

P Douglas Boatman, Brett Lauring, Thomas O Schrader, Michelle Kasem, Benjamin R Johnson, Philip Skinner, Jae-Kyu Jung, Jerry Xu, Martin C Cherrier, Peter J Webb, Graeme Semple, Carleton R Sage, Jens Knudsen, Ruoping Chen, Wen-Lin Luo, Luzelena Caro, Josee Cote, Eseng Lai, John Wagner, Andrew K Tagga

Crystal structure of the human spastin AAA domain

人类 Spastin AAA 结构域的晶体结构

Jennifer L Taylor, Susan Roehl White, Brett Lauring, F Jon Kull