INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology
INCB24360(Epacadostat),一种高效且选择性的吲哚胺-2,3-双加氧酶1(IDO1)抑制剂,用于免疫肿瘤学
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.6b00391
Yue, Eddy W; Sparks, Richard; Polam, Padmaja; Modi, Dilip; Douty, Brent; Wayland, Brian; Glass, Brian; Takvorian, Amy; Glenn, Joseph; Zhu, Wenyu; Bower, Michael; Liu, Xiangdong; Leffet, Lynn; Wang, Qian; Bowman, Kevin J; Hansbury, Michael J; Wei, Min; Li, Yanlong; Wynn, Richard; Burn, Timothy C; Koblish, Holly K; Fridman, Jordan S; Emm, Tom; Scherle, Peggy A; Metcalf, Brian; Combs, Andrew P