Discovery of INCB126503 as a Potent and Selective FGFR2/3 Inhibitor
发现 INCB126503 是一种高效且选择性的 FGFR2/3 抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00232
Nguyen, Minh H; Wang, Anlai; Truong, Lisa; Zhang, Ke; Ye, Hai-Fen; Zhao, Peng; Horsey, April; Frascella, Michelle; Leffet, Lynn; Federowicz, Kelly; Behshad, Elham; Witten, Michael R; Qi, Chao; Xu, Yao; Jalluri, Ravi; Harris, Jennifer J; Hess, Rodrigo; Sayers, Brian; Lin, Luping; Yeleswaram, Swamy; Zhang, Guofeng; Kim, Sunkyu; Covington, Maryanne; Diamond, Sharon; Yao, Wenqing; Vechorkin, Oleg