Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit
通过优化片段匹配来识别 VIII 家族溴结构域的化学探针
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.6b00012
Brian S Gerstenberger, John D Trzupek, Cynthia Tallant, Oleg Fedorov, Panagis Filippakopoulos, Paul E Brennan, Vita Fedele, Sarah Martin, Sarah Picaud, Catherine Rogers, Mihir Parikh, Alexandria Taylor, Brian Samas, Alison O'Mahony, Ellen Berg, Gabriel Pallares, Adam D Torrey, Daniel K Treiber, Ivan
