Development of new scaffolds as reversible tissue transglutaminase inhibitors, with improved potency or resistance to glutathione addition
开发新型支架作为可逆性组织转谷氨酰胺酶抑制剂,以提高其效力或对谷胱甘肽添加的耐受性
期刊:Medchemcomm
影响因子:
doi:10.1039/c6md00565a
Apperley, Kim Y P; Roy, Isabelle; Saucier, Vincent; Brunet-Filion, Nicholas; Piscopo, Sara-Pier; Pardin, Christophe; De Francesco, Élise; Hao, Catherine; Keillor, Jeffrey W