日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Thiadiazolopyrimidinone-Based Molecule Targeting Annexin A6 Impairs Cell Motility and Epithelial-to-Mesenchymal Transition in Pancreatic Cancer Cells Lacking Annexin A1

一种靶向 Annexin A6 的噻二唑并嘧啶酮类分子可抑制缺乏 Annexin A1 的胰腺癌细胞的运动性和上皮间质转化。

Belvedere, Raffaella; Novizio, Nunzia; Ruggiero, Dafne; Palazzo, Mariangela; Bruno, Ines; Terracciano, Stefania; Petrella, Antonello

From Bench to Bedside: Translational Approaches to Cardiotoxicity in Breast Cancer, Lung Cancer, and Lymphoma Therapies

从实验室到临床:乳腺癌、肺癌和淋巴瘤治疗中心脏毒性的转化研究

Nardone, Valerio; Ruggiero, Dafne; Chini, Maria Giovanna; Bruno, Ines; Lauro, Gianluigi; Terracciano, Stefania; Nebbioso, Angela; Bifulco, Giuseppe; Cappabianca, Salvatore; Reginelli, Alfonso

Identification of a New Interesting BAG3 Modulator Able to Disrupt Cancer-Related Pathways

鉴定出一种能够干扰癌症相关通路的新型有趣的BAG3调节剂

Ruggiero, Dafne; Boccia, Eleonora; Ingenito, Emis; Vestuto, Vincenzo; D'Urso, Gilda; Capuano, Alessandra; Casapullo, Agostino; Terracciano, Stefania; Bifulco, Giuseppe; Lauro, Gianluigi; Bruno, Ines

Unveiling New Triazoloquinoxaline-Based PROTACs Designed for the Selective Degradation of the ncBAF Chromatin Remodeling Subunit BRD9.

推出新型三唑喹喔啉基 PROTAC,用于选择性降解 ncBAF 染色质重塑亚基 BRD9

Pierri Martina, Bove Guglielmo, Gazzillo Erica, Colarusso Ester, Scala Francesca, Pepe Giacomo, Terracciano Stefania, Chini Maria Giovanna, Simonelli Nicla, Bruno Ines, Nebbioso Angela, Campiglia Pietro, Bifulco Giuseppe, Altucci Lucia, Del Gaudio Nunzio, Lauro Gianluigi

Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E(2) and Leukotriene Biosynthesis Inhibitors

鉴定2-氨基酰基-1,3,4-噻二唑类化合物为前列腺素E(2)和白三烯生物合成抑制剂

Potenza, Marianna; Giordano, Assunta; Chini, Maria G; Saviano, Anella; Kretzer, Christian; Raucci, Federica; Russo, Marina; Lauro, Gianluigi; Terracciano, Stefania; Bruno, Ines; Iorizzi, Maria; Hofstetter, Robert K; Pace, Simona; Maione, Francesco; Werz, Oliver; Bifulco, Giuseppe

Identification of 2,4-Dinitro-Biphenyl-Based Compounds as MAPEG Inhibitors

鉴定2,4-二硝基联苯类化合物作为MAPEG抑制剂

Di Micco, Simone; Terracciano, Stefania; Pierri, Martina; Cantone, Vincenza; Liening, Stefanie; König, Stefanie; Garscha, Ulrike; Hofstetter, Robert Klaus; Koeberle, Andreas; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe

Targeting mPGES-1 by a Combinatorial Approach: Identification of the Aminobenzothiazole Scaffold to Suppress PGE(2) Levels

通过组合策略靶向 mPGES-1:鉴定氨基苯并噻唑骨架以抑制 PGE(2) 水平

Chini, Maria G; Giordano, Assunta; Potenza, Marianna; Terracciano, Stefania; Fischer, Katrin; Vaccaro, Maria C; Colarusso, Ester; Bruno, Ines; Riccio, Raffaele; Koeberle, Andreas; Werz, Oliver; Bifulco, Giuseppe

Identification of the 2-Benzoxazol-2-yl-phenol Scaffold as New Hit for JMJD3 Inhibition

鉴定出 2-苯并恶唑-2-基苯酚骨架为 JMJD3 抑制剂的新先导化合物

Giordano, Assunta; Forte, Giovanni; Terracciano, Stefania; Russo, Alessandra; Sala, Marina; Scala, Maria C; Johansson, Catrine; Oppermann, Udo; Riccio, Raffaele; Bruno, Ines; Di Micco, Simone