CC4, a dimer of cytisine, is a selective partial agonist at α4β2/α6β2 nAChR with improved selectivity for tobacco smoking cessation
CC4 是金雀花碱的二聚体,是 α4β2/α6β2 nAChR 的选择性部分激动剂,对戒烟具有更高的选择性
期刊:British Journal of Pharmacology
影响因子:6.8
doi:10.1111/j.1476-5381.2012.02204.x
Mariaelvina Sala, Daniela Braida, Luca Pucci, Irene Manfredi, Michael J Marks, Charles R Wageman, Sharon R Grady, Barbara Loi, Sergio Fucile, Francesca Fasoli, Michele Zoli, Bruno Tasso, Fabio Sparatore, Francesco Clementi, Cecilia Gotti