日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Investigations of Antioxidant and Anti-Cancer Activities of 5-Aminopyrazole Derivatives

5-氨基吡唑衍生物抗氧化及抗癌活性研究

Federica Rapetti, Andrea Spallarossa, Eleonora Russo, Debora Caviglia, Carla Villa, Bruno Tasso, Maria Grazia Signorello, Camillo Rosano, Erika Iervasi, Marco Ponassi, Chiara Brullo

Discovery of Novel Thiazole-Based SIRT2 Inhibitors as Anticancer Agents: Molecular Modeling, Chemical Synthesis and Biological Assays

发现新型噻唑类 SIRT2 抑制剂作为抗癌剂:分子建模、化学合成和生物测定

Francesco Piacente, Giorgia Guccione, Naomi Scarano, Dario Lunaccio, Caterina Miro, Elena Abbotto, Annalisa Salis, Bruno Tasso, Monica Dentice, Santina Bruzzone, Elena Cichero, Enrico Millo

PTC596-Induced BMI-1 Inhibition Fights Neuroblastoma Multidrug Resistance by Inducing Ferroptosis

PTC596 诱导的 BMI-1 抑制通过诱导铁死亡来对抗神经母细胞瘤多药耐药性

Giulia Elda Valenti, Antonella Roveri, Rina Venerando, Paola Menichini, Paola Monti, Bruno Tasso, Nicola Traverso, Cinzia Domenicotti, Barbara Marengo

Journey on VX-809-Based Hybrid Derivatives towards Drug-like F508del-CFTR Correctors: From Molecular Modeling to Chemical Synthesis and Biological Assays

基于 VX-809 的混合衍生物向类药物 F508del-CFTR 校正剂的演进:从分子建模到化学合成和生物测定

Alice Parodi, Giada Righetti, Emanuela Pesce, Annalisa Salis, Valeria Tomati, Cristina Pastorino, Bruno Tasso, Mirko Benvenuti, Gianluca Damonte, Nicoletta Pedemonte, Elena Cichero, Enrico Millo

Multitarget Biological Profiling of New Naphthoquinone and Anthraquinone-Based Derivatives for the Treatment of Alzheimer's Disease

用于治疗阿尔茨海默病的新型萘醌和蒽醌基衍生物的多靶点生物学分析

Marta Campora, Claudio Canale, Elena Gatta, Bruno Tasso, Erik Laurini, Annalisa Relini, Sabrina Pricl, Marco Catto, Michele Tonelli

CC4, a dimer of cytisine, is a selective partial agonist at α4β2/α6β2 nAChR with improved selectivity for tobacco smoking cessation

CC4 是金雀花碱的二聚体,是 α4β2/α6β2 nAChR 的选择性部分激动剂,对戒烟具有更高的选择性

Mariaelvina Sala, Daniela Braida, Luca Pucci, Irene Manfredi, Michael J Marks, Charles R Wageman, Sharon R Grady, Barbara Loi, Sergio Fucile, Francesca Fasoli, Michele Zoli, Bruno Tasso, Fabio Sparatore, Francesco Clementi, Cecilia Gotti

Antiviral and cytotoxic activities of aminoarylazo compounds and aryltriazene derivatives

氨基芳基偶氮化合物和芳基三氮烯衍生物的抗病毒和细胞毒活性

Michele Tonelli, Iana Vazzana, Bruno Tasso, Vito Boido, Fabio Sparatore, Maurizio Fermeglia, Maria Silvia Paneni, Paola Posocco, Sabrina Pricl, Paolo La Colla, Cristina Ibba, Barbara Secci, Gabriella Collu, Roberta Loddo