日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Design of PROTACS for the Degradation of Soluble Epoxide Hydrolase.

基于结构的PROTACS设计用于降解可溶性环氧化物水解酶

Schönfeld Julia, Brunst Steffen, Ciomirtan Ludmila, Willmer Lena, Chromik Michel A, Kumar Adarsh, Froemel Timo, Liebisch Nick, Hackspacher Arne, Ehrler Johanna H M, Wintermeier Lukas, Hesse Christina, Fiedler Jan, Heering Jan, Freitag Hinrich, Zardo Patrick, Fieguth Hans-Gerd, Brüggerhoff Astrid, Jakob Josefine, Häupl Björn, Weizel Lilia, Kaiser Astrid, Schubert-Zsilavecz Manfred, Oellerich Thomas, Fleming Ingrid, Schebb Nils H, Fürst Robert, Kannt Aimo, Knapp Stefan, Proschak Ewgenij, Hiesinger Kerstin

Sustainable Joullié-Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors.

可持续的 Joullié-Ugi 和连续流实施产生了新型的受卡托普利启发的广谱金属β-内酰胺酶抑制剂

Alfano Antonella Ilenia, Pelliccia Sveva, Barone Simona, Cutarella Luigi, Cancade Sacha Michèle Idriss, Baia Valerio, Cassese Emilia, Russomanno Pasquale, Messano Nicolò, Frank Denia, Weizel Lilia, Rotter Marco J, Brunst Steffen, Wichelhaus Thomas A, Proschak Ewgenij, Tedesco Daniele, Mori Mattia, Docquier Jean Denis, Summa Vincenzo, Brindisi Margherita

Designing a Small Fluorescent Inhibitor to Investigate Soluble Epoxide Hydrolase Engagement in Living Cells

设计一种小型荧光抑制剂来研究活细胞中可溶性环氧化物水解酶的活性

Brunst, Steffen; Schönfeld, Julia; Breunig, Peter; Burgers, Luisa D; DeMeglio, Murphy; Ehrler, Johanna H M; Lillich, Felix F; Weizel, Lilia; Hefendehl, Jasmin K; Fürst, Robert; Proschak, Ewgenij; Hiesinger, Kerstin

Rh(II) -Catalyzed De-symmetrization of Ethane-1,2-dithiol and Propane-1,3-dithiol Yields Metallo-β-lactamase Inhibitors

Rh(II)催化乙烷-1,2-二硫醇和丙烷-1,3-二硫醇的去对称化反应生成金属β-内酰胺酶抑制剂

Krasavin, Mikhail; Zhukovsky, Daniil; Solovyev, Igor; Barkhatova, Darina; Dar'in, Dmitry; Frank, Denia; Martinelli, Giada; Weizel, Lilia; Proschak, Anna; Rotter, Marco; Kramer, Jan S; Brunst, Steffen; Wichelhaus, Thomas A; Proschak, Ewgenij

Development and in vitro Profiling of Dual FXR/LTA4H Modulators

双重FXR/LTA4H调节剂的开发和体外特性分析

Schierle, Simone; Brunst, Steffen; Helmstädter, Moritz; Ebert, Roland; Kramer, Jan S; Steinhilber, Dieter; Proschak, Ewgenij; Merk, Daniel

Systematic Assessment of Fragment Identification for Multitarget Drug Design

多靶点药物设计中片段识别的系统性评估

Brunst, Steffen; Kramer, Jan S; Kilu, Whitney; Heering, Jan; Pollinger, Julius; Hiesinger, Kerstin; George, Sven; Steinhilber, Dieter; Merk, Daniel; Proschak, Ewgenij