日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

PAC1 receptor blockade reduces central nociceptive activity: new approach for primary headache?

PAC1 受体阻断可降低中枢伤害感受活动:治疗原发性头痛的新方法?

Jan Hoffmann, Silke Miller, Margarida Martins-Oliveira, Simon Akerman, Weera Supronsinchai, Hong Sun, Licheng Shi, Judy Wang, Dawn Zhu, Sonya Lehto, Hantao Liu, Ruoyuan Yin, Bryan D Moyer, Cen Xu, Peter J Goadsby

Pharmacological characterization of potent and selective NaV1.7 inhibitors engineered from Chilobrachys jingzhao tarantula venom peptide JzTx-V

以 Chilobrachys jingzhao 狼蛛毒肽 JzTx-V 为原料,设计出强效、选择性 NaV1.7 抑制剂的药理学特性

Bryan D Moyer, Justin K Murray, Joseph Ligutti, Kristin Andrews, Philippe Favreau, John B Jordan, Josie H Lee, Dong Liu, Jason Long, Kelvin Sham, Licheng Shi, Reto Stöcklin, Bin Wu, Ruoyuan Yin, Violeta Yu, Anruo Zou, Kaustav Biswas, Les P Miranda

Evaluation of recombinant monoclonal antibody SVmab1 binding to Na V1.7 target sequences and block of human Na V1.7 currents

评估重组单克隆抗体 SVmab1 与 Na V1.7 靶序列结合并阻断人类 Na V1.7 电流

Dong Liu, Mandy Tseng, Linda F Epstein, Lydia Green, Brian Chan, Brian Soriano, Desiree Lim, Oscar Pan, Christopher M Murawsky, Chadwick T King, Bryan D Moyer

Voltage-gated sodium channels in taste bud cells

味蕾细胞中的电压门控钠通道

Na Gao, Min Lu, Fernando Echeverri, Bianca Laita, Dalia Kalabat, Mark E Williams, Peter Hevezi, Albert Zlotnik, Bryan D Moyer