日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-based design of an opioid receptor modulator for enhanced morphine analgesia

基于结构的阿片受体调节剂设计及其在增强吗啡镇痛中的应用

Wang, Yue; Luo, Ping; Xu, Haiyan; Zhan, Li; Sakamoto, Kensuke; Li, Mingyu; Wang, Jing; Huang, Xi-Ping; Zhou, Jianhui; Liu, Tao; Suo, Yanrui; Fan, Wenjia; He, Xinheng; Xu, Youwei; Cai, Yongjie; Wang, Chao; Zhao, Yuxi; Dai, Antao; Lai, Yali; Yuan, Qingning; Hu, Wen; Wu, Kai; Yang, Dehua; Cheng, Xi; Lu, Xiaojie; Krumm, Brian; Kenakin, Terry; Zhang, Jian; Roth, Bryan L; Gao, Zhaobing; Xu, H Eric; Zhuang, Youwen

Structural insights into coffee bitter taste perception by TAS2R43 receptor

TAS2R43受体对咖啡苦味感知的结构性见解

Kim, Yoojoong; Gumpper, Ryan H; Zhuang, Yuxuan; Dror, Ron O; Roth, Bryan L

Large Library Docking for Polypharmacology

用于多药理学的大型库对接

Wu, Yujin; Vigneron, Seth; Braz, Joao; Srinivasan, Karthik; Fink, Elissa A; Huang, Xi-Ping; Xu, Xinyu; Huebner, Harald; Kim, Joseph Y; Wang, Jing; Pfeiffer, Tara; Sakamoto, Kensuke; Radchenko, Dmytro S; Rodriguiz, Ramona M; Moroz, Yurii S; Irwin, John J; Gmeiner, Peter; Billesboelle, Christian; Roth, Bryan L; Basbaum, Allan I; Manglik, Aashish; Wetsel, William C; Shoichet, Brian K

A Defined Patho-Mechanism for Acute Radiation Syndrome Death and a Three-Drug Regimen to Prevent It

急性放射综合征死亡的明确病理机制及预防该疾病的三药方案

Fahl, William E; Goesch, Hannah R; Goesch, Sarah R; Fahl, Bryan L

Temporal molecular remodeling of T cells informs their possible adaptation in 4T1 tumors

T细胞的分子重塑的时间性变化揭示了它们在4T1肿瘤中可能的适应性

Iftehimul, Md; Newman, Robert H; Harrison, Scott H; Jones, Roshonda B; Muganda, Perpetua M; Holloman, Bryan L; Hossain, Muhammad T; Rorie, Checo J; Thomas, Misty D; Graves, Joseph L Jr; Kaufman, Howard L; Saha, Dipongkor

Effect of Liver Metastases on Survival in Microsatellite-Stable Metastatic Colorectal Cancer Treated with Immune Checkpoint Inhibitors

肝转移对接受免疫检查点抑制剂治疗的微卫星稳定型转移性结直肠癌患者生存的影响

Pakvisal, Nussara; Pappas, Leontios; Caughey, Bennett A; Horick, Nora K; Tarazona, Noelia; Vora, Kruti B; Ouyang, Ben; Pandey, Aditya; Peacker, Bryan L; Sun, Joie; Zubiri, Leyre; Reynolds, Kerry L; Ryan, David P; Qadan, Motaz; Corcoran, Ryan B; Giantonio, Bruce; Allen, Jill N; Walsh, Elizabeth P; Clark, Jefferey W; Ting, David T; Parikh, Aparna R

A new sensitive derivatization assay of PrC-210 in plasma and tissues using liquid chromatography coupled with tandem mass spectrometry

利用液相色谱-串联质谱法测定血浆和组织中 PrC-210 的新型高灵敏度衍生化方法

Fahl, Bryan L; Scarlett, Cameron O; Fahl, William E

Multidisciplinary Approach to Complex Lower Extremity Limb Salvage in Pyogenic Arthritis, Pyoderma Gangrenosum, and Acne (PAPA) Syndrome: A Case Report

化脓性关节炎、坏疽性脓皮病和痤疮(PAPA)综合征复杂下肢肢体挽救的多学科治疗方法:病例报告

Talanker, Michael M; Basta, Anthony V; Do, Tien; Tung, Robert; Allen, Addison; Martin, Morgan; Ruygrok, Bryan L; Kellam, Patrick J; Trost, Jeffrey G; Bhadkamkar, Mohin A

Cryo-EM Structures of Brain-Derived G Protein-Coupled Receptors: The First Direct Visualization from Mammalian Brain Tissue

脑源性G蛋白偶联受体的冷冻电镜结构:首次从哺乳动物脑组织中直接观察

Wright, Nicholas J; Chiu, Yi-Ting; Sakamoto, Kensuke; Kocak, D Dewran; Fordyce, Blake A; Hua, Kunjie; Huang, Karen Lu; Scherrer, Grégory; Lyons, Scott P; Roth, Bryan L

Xylazine's κ opioid agonist activity is not shared with other FDA-approved α(2)-adrenergic agonists

赛拉嗪的κ阿片受体激动剂活性与其他FDA批准的α(2)-肾上腺素能激动剂不同。

Huang, Xi-Ping; Krumm, Brian E; Bedard, Madigan L; McElligott, Zoe A; Roth, Bryan L