日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting carbonic anhydrase IX/XII prevents the anti-ferroptotic effect of stromal lactic acid in prostate carcinoma.

靶向碳酸酐酶 IX/XII 可阻止基质乳酸在前列腺癌中的抗铁死亡作用

Pardella Elisa, Comito Giuseppina, Ippolito Luigi, Pranzini Erica, Iozzo Marta, Gangarossa Giulia, Virgilio Francesca, Bua Silvia, Nocentini Alessio, Sandrini Giada, Lorito Nicla, Bacci Marina, Nesi Gabriella, Spatafora Pietro, Serni Sergio, Supuran Claudiu T, Morandi Andrea, Chiarugi Paola, Giannoni Elisa

Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae.

针对耐多药淋病奈瑟菌的青霉素类碳酸酐酶抑制剂的研发

Bonardi Alessandro, Nocentini Alessio, Giovannuzzi Simone, Paoletti Niccolò, Ammara Andrea, Bua Silvia, Abutaleb Nader S, Abdelsattar Abdallah S, Capasso Clemente, Gratteri Paola, Flaherty Daniel P, Seleem Mohamed N, Supuran Claudiu T

Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains

苯并噻二嗪酮-1,1-二氧化物碳酸酐酶抑制剂可抑制耐药结核分枝杆菌菌株的生长

Bua, Silvia; Bonardi, Alessandro; Mük, Georgiana Ramona; Nocentini, Alessio; Gratteri, Paola; Supuran, Claudiu T

Carbonic anhydrase inhibitory activity of phthalimide-capped benzene sulphonamide derivatives

邻苯二甲酰亚胺封端的苯磺酰胺衍生物的碳酸酐酶抑制活性

Shilkar, Deepak; Mohd Siddique, Mohd Usman; Bua, Silvia; Yasmin, Sabina; Patil, Mrunali; Timiri, Ajay Kumar; Supuran, Claudiu T; Jayaprakash, Venkatesan

Design, synthesis, and carbonic anhydrase inhibition activities of Schiff bases incorporating benzenesulfonamide scaffold: Molecular docking application

含苯磺酰胺骨架的席夫碱的设计、合成及其碳酸酐酶抑制活性:分子对接应用

El-Azab, Adel S; A-M Abdel-Aziz, Alaa; Bua, Silvia; Nocentini, Alessio; Bakheit, Ahmed H; Alkahtani, Hamad M; Hefnawy, Mohamed M; Supuran, Claudiu T

Toxicity evaluation of sulfamides and coumarins that efficiently inhibit human carbonic anhydrases

有效抑制人碳酸酐酶的磺胺类和香豆素类化合物的毒性评价

Aspatwar, Ashok; Berrino, Emanuela; Bua, Silvia; Carta, Fabrizio; Capasso, Clemente; Parkkila, Seppo; Supuran, Claudiu T

Escherichia coli γ-carbonic anhydrase: characterisation and effects of simple aromatic/heterocyclic sulphonamide inhibitors

大肠杆菌γ-碳酸酐酶:简单芳香族/杂环磺酰胺抑制剂的特性及作用

Del Prete, Sonia; Bua, Silvia; Supuran, Claudiu T; Capasso, Clemente

Dual P-Glycoprotein and CA XII Inhibitors: A New Strategy to Reverse the P-gp Mediated Multidrug Resistance (MDR) in Cancer Cells

双重P-糖蛋白和CA XII抑制剂:逆转癌细胞P-gp介导的多药耐药性(MDR)的新策略

Teodori, Elisabetta; Braconi, Laura; Bua, Silvia; Lapucci, Andrea; Bartolucci, Gianluca; Manetti, Dina; Romanelli, Maria Novella; Dei, Silvia; Supuran, Claudiu T; Coronnello, Marcella

Comparison of the Sulfonamide Inhibition Profiles of the α-Carbonic Anhydrase Isoforms (SpiCA1, SpiCA2 and SpiCA3) Encoded by the Genome of the Scleractinian Coral Stylophora pistillata

对石珊瑚 Stylophora pistillata 基因组编码的 α-碳酸酐酶同工酶(SpiCA1、SpiCA2 和 SpiCA3)的磺胺类药物抑制谱进行比较

Del Prete, Sonia; Bua, Silvia; Alasmary, Fatmah A S; AlOthman, Zeid; Tambutté, Sylvie; Zoccola, Didier; Supuran, Claudiu T; Capasso, Clemente

Novel 8-Substituted Coumarins That Selectively Inhibit Human Carbonic Anhydrase IX and XII

新型8-取代香豆素选择性抑制人碳酸酐酶IX和XII

Buran, Kerem; Bua, Silvia; Poli, Giulio; Önen Bayram, F Esra; Tuccinardi, Tiziano; Supuran, Claudiu T