日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

WRN structural flexibility showcased through fragment-based lead discovery of inhibitors

通过基于片段的抑制剂先导化合物发现,展现了WRN结构的灵活性

Palte, Rachel L; Mandal, Mihir; Sikorska, Justyna; Villafania, Artjohn B; Rickard, Meredith M; Bauer, Robert J; Buevich, Alexei V; Chai, Xiaomei; He, Jiafang; Hussain, Zahid; Koglin, Markus; MacDonald, Hannah B; Mansueto, My S; Maskos, Klaus; Methot, Joey L; Robustelli, Jaclyn; Soriano, Aileen; Tauchert, Marcel J; Tyagarajan, Sriram; Zhang, Minjia; Klein, Daniel J; Hicks, Jacqueline D; McLaren, David G; Gabelli, Sandra B; Wyss, Daniel F

Rapid Affinity and Microsomal Stability Ranking of Crude Mixture Libraries of Histone Deacetylase Inhibitors

组蛋白去乙酰化酶抑制剂粗提物库的快速亲和力和微粒体稳定性排序

Tyagarajan, Sriram; Andrews, Christine L; Beshore, Douglas C; Buevich, Alexei V; Curran, Patrick J; Dandliker, Peter; Greshock, Thomas J; Hoar, Jason; Kim, Alex; Karnachi, Prabha; Knemeyer, Ian; Kozlowski, Joseph; Liu, Jian; Maletic, Milana; Myers, Robert; Rada, Vanessa; Sha, Deyou; Sauvagnat, Berengere; Vachal, Petr; Wolkenberg, Scott; Yu, Wensheng; Yu, Younong; Krska, Shane W

DELTA50: A Highly Accurate Database of Experimental (1)H and (13)C NMR Chemical Shifts Applied to DFT Benchmarking

DELTA50:一个高精度的实验(1)H和(13)C NMR化学位移数据库,应用于DFT基准测试

Cohen, Ryan D; Wood, Jared S; Lam, Yu-Hong; Buevich, Alexei V; Sherer, Edward C; Reibarkh, Mikhail; Williamson, R Thomas; Martin, Gary E

Enhancing Efficiency of Natural Product Structure Revision: Leveraging CASE and DFT over Total Synthesis

提高天然产物结构修正效率:利用CASE和DFT方法改进全合成

Elyashberg, Mikhail; Tyagarajan, Sriram; Mandal, Mihir; Buevich, Alexei V

Ominoxanthone-The First Xanthone Linearly Fused to a γ-Lactone from Cortinarius ominosus Bidaud Basidiomata. CASE- and DFT-Based Structure Elucidation

Ominoxanthone - 第一个线性融合到 Cortinarius ominosus Bidaud Basidiomata 的 γ-内酯上的 Xanthone。基于 CASE 和 DFT 的结构解析

Alice Trac, Célia Issaad, Mehdi A Beniddir, Jean-Michel Bellanger, Jean-François Gallard, Alexei V Buevich, Mikhail E Elyashberg, Pierre Le Pogam

Photoredox-Catalyzed Giese Reactions: Decarboxylative Additions to Cyclic Vinylogous Amides and Esters

光氧化还原催化吉斯反应:环状乙烯基酰胺和酯的脱羧加成反应

Dykstra, Kevin; Buevich, Alexei; Gao, Qi; Lam, Yu-Hong; Kuethe, Jeffrey T

Acupuncture in the Treatment of Sequestered Intervertebral Disk Herniation

针灸治疗游离型椎间盘突出症

Buevich, Vadim; Buevich, Maxim; Buevich, Natalia

An orally available non-nucleotide STING agonist with antitumor activity

一种具有抗肿瘤活性的口服非核苷酸 STING 激动剂

Bo-Sheng Pan #, Samanthi A Perera #, Jennifer A Piesvaux #, Jeremy P Presland #, Gottfried K Schroeder #, Jared N Cumming #, B Wesley Trotter #, Michael D Altman, Alexei V Buevich, Brandon Cash, Saso Cemerski, Wonsuk Chang, Yiping Chen, Peter J Dandliker, Guo Feng, Andrew Haidle, Timothy Henderson, 

An Open-Label Extension Study to Assess the Long-Term Efficacy and Safety of a Plasma-Derived von Willebrand Factor (VWF)/Factor VIII (FVIII) Concentrate in Patients with von Willebrand Disease (SWIFT-VWDext Study)

一项开放标签扩展研究,旨在评估血浆来源的血管性血友病因子 (VWF)/因子 VIII (FVIII) 浓缩物在血管性血友病患者中的长期疗效和安全性 (SWIFT-VWDext 研究)

Lissitchkov, Toshko; Klukowska, Anna; Buevich, Evgeny; Maltceva, Irina; Auerswald, Guenter; Stasyshyn, Oleksandra; Seifert, Wilfried; Rogosch, Tobias

MK-8353: Discovery of an Orally Bioavailable Dual Mechanism ERK Inhibitor for Oncology

MK-8353:一种用于肿瘤治疗的口服生物利用度高的双机制ERK抑制剂的发现

Boga, Sobhana Babu; Deng, Yongqi; Zhu, Liang; Nan, Yang; Cooper, Alan B; Shipps, Gerald W Jr; Doll, Ronald; Shih, Neng-Yang; Zhu, Hugh; Sun, Robert; Wang, Tong; Paliwal, Sunil; Tsui, Hon-Chung; Gao, Xiaolei; Yao, Xin; Desai, Jagdish; Wang, James; Alhassan, Abdul Basit; Kelly, Joseph; Patel, Mehul; Muppalla, Kiran; Gudipati, Subrahmanyam; Zhang, Li-Kang; Buevich, Alexei; Hesk, David; Carr, Donna; Dayananth, Priya; Black, Stuart; Mei, Hong; Cox, Kathleen; Sherborne, Bradley; Hruza, Alan W; Xiao, Li; Jin, Weihong; Long, Brian; Liu, Gongjie; Taylor, Stacey A; Kirschmeier, Paul; Windsor, William T; Bishop, Robert; Samatar, Ahmed A