Discovery and SAR of Novel 2,3-Dihydroimidazo[1,2-c]quinazoline PI3K Inhibitors: Identification of Copanlisib (BAY 80-6946)
新型 2,3-二氢咪唑并[1,2-c]喹唑啉 PI3K 抑制剂的发现和构效关系研究:Copanlisib (BAY 80-6946) 的鉴定
期刊:ChemMedChem
影响因子:3.4
doi:10.1002/cmdc.201600148
Scott, William J; Hentemann, Martin F; Rowley, R Bruce; Bull, Cathy O; Jenkins, Susan; Bullion, Ann M; Johnson, Jeffrey; Redman, Anikó; Robbins, Arthur H; Esler, William; Fracasso, R Paul; Garrison, Timothy; Hamilton, Mark; Michels, Martin; Wood, Jill E; Wilkie, Dean P; Xiao, Hong; Levy, Joan; Stasik, Enrico; Liu, Ningshu; Schaefer, Martina; Brands, Michael; Lefranc, Julien