日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Binding kinetics, bias, receptor internalization and effects on insulin secretion in vitro and in vivo of a novel GLP-1R/GIPR dual agonist, HISHS-2001

新型 GLP-1R/GIPR 双重激动剂 HISHS-2001 的结合动力学、偏向性、受体内化及其对体外和体内胰岛素分泌的影响

Yusman Manchanda ,Ben Jones ,Gaelle Carrat ,Zenouska Ramchunder ,Piero Marchetti ,Isabelle Leclerc ,Rajamannar Thennati ,Vinod Burade ,Muthukumaran Natarajan ,Pradeep Shahi ,Alejandra Tomas ,Guy A Rutter

Assessing Change in Stone Burden on Baseline and Follow-Up CT: Radiologist and Radiomics Evaluations

评估基线和随访CT扫描中结石负荷的变化:放射科医生和放射组学评估

Kaviani, Parisa; Froelich, Matthias F; Bizzo, Bernardo; Primak, Andrew; Dasegowda, Giridhar; Garza-Frias, Emiliano; Karout, Lina; Burade, Anushree; Hosseini, Seyedehelaheh; Contreras Yametti, Javier Eduardo; Dreyer, Keith; Saini, Sanjay; Kalra, Mannudeep

Binding Kinetics, Bias, Receptor Internalization and Effects on Insulin Secretion in vitro and in vivo of a Novel GLP-1R/GIPR Dual Agonist, HISHS-2001

新型 GLP-1R/GIPR 双重激动剂的结合动力学、偏差、受体内化以及对体内和体外胰岛素分泌的影响,HISHS-2001

Yusman Manchanda, Ben Jones, Gaelle Carrat, Zenouska Ramchunder, Piero Marchetti, Isabelle Leclerc, Rajamannar Thennati, Vinod Burade, Muthukumaran Natarajan, Pradeep Shahi, Alejandra Tomas, Guy A Rutter

2-Deoxy-4-epi-scyllo-inosose (DEI) is the Product of EboD, a Highly Conserved Dehydroquinate Synthase-like Enzyme in Bacteria and Eustigmatophyte Algae

2-脱氧-4-表-肌醇糖(DEI)是EboD的产物,EboD是细菌和真眼点藻类中高度保守的脱氢奎宁酸合酶样酶。

Tanoeyadi, Samuel; Zhou, Wei; Osborn, Andrew R; Tsunoda, Takeshi; Samadi, Arash; Burade, Sachin; Waldo, Ty J; Higgins, Melanie A; Mahmud, Taifo

Complete biosynthetic pathway to the antidiabetic drug acarbose

抗糖尿病药物阿卡波糖的完整生物合成途径

Takeshi Tsunoda, Arash Samadi, Sachin Burade, Taifo Mahmud

In vivo and in vitro characterization of GL0034, a novel long-acting glucagon-like peptide-1 receptor agonist

新型长效胰高血糖素样肽-1受体激动剂GL0034的体内和体外表征

Ben Jones, Vinod Burade, Elina Akalestou, Yusman Manchanda, Zenouska Ramchunder, Gaëlle Carrat, Marie-Sophie Nguyen-Tu, Piero Marchetti, Lorenzo Piemonti, Isabelle Leclerc, Rajamannar Thennati, Tina Vilsboll, Bernard Thorens, Alejandra Tomas, Guy A Rutter

Preclinical Efficacy Comparison of Cyclosporine Ophthalmic Solution 0.09% vs Cyclosporine Ophthalmic Emulsion 0.05% vs Ciclosporin Ophthalmic Emulsion 0.1% in a NOD Mouse Model of Dry Eye Disease

0.09% 环孢素眼用溶液、0.05% 环孢素眼用乳剂和 0.1% 环孢素眼用乳剂在 NOD 小鼠干眼症模型中的临床前疗效比较

Vinod Burade, Rishit Zalawadia, Alpesh Patel, Abayomi Ogundele

Analytical characterization of recombinant hCG and comparative studies with reference product

重组 hCG 的分析表征及与参比产品的比较研究

Rajamannar Thennati, Sanjay Kumar Singh, Nitin Nage, Yena Patel, Sandip Kumar Bose, Vinod Burade, Ranjit Sudhakar Ranbhor

Comparative plasma and tissue distribution of Sun Pharma's generic doxorubicin HCl liposome injection versus Caelyx(®) (doxorubicin HCl liposome injection) in syngeneic fibrosarcoma-bearing BALB/c mice and Sprague-Dawley rats

在同源纤维肉瘤BALB/c小鼠和Sprague-Dawley大鼠中,Sun Pharma的仿制药盐酸阿霉素脂质体注射液与Caelyx(®)(盐酸阿霉素脂质体注射液)的血浆和组织分布比较

Burade, Vinod; Bhowmick, Subhas; Maiti, Kuntal; Zalawadia, Rishit; Jain, Deepak; Rajamannar, Thennati