日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Taurine-Based Hybrid Drugs as Potential Anticancer Therapeutic Agents: In Vitro, In Vivo Evaluations.

牛磺酸基混合药物作为潜在的抗癌治疗剂:体外、体内评价

Nakypova Saltanat, Smolobochkin Andrey, Rizbayeva Tanzilya, Turmanov Rakhymzhan, Gazizov Almir, Akylbekov Nurgali, Zhapparbergenov Rakhmetulla, Narmanova Roza, Ibadullayeva Saltanat, Zalaltdinova Alena, Syzdykbayev Marat, Voronina Julia, Lyubina Anna, Voloshina Alexandra, Klimanova Elena, Sashenkova Tatiana, Mishchenko Denis, Burilov Alexander

Progress in the Stereoselective Synthesis Methods of Pyrrolidine-Containing Drugs and Their Precursors

含吡咯烷药物及其前体的立体选择性合成方法的研究进展

Smolobochkin, Andrey; Gazizov, Almir; Appazov, Nurbol; Sinyashin, Oleg; Burilov, Alexander

Superelectrophilic Activation of Phosphacoumarins towards Weak Nucleophiles via Brønsted Acid Assisted Brønsted Acid Catalysis

布朗斯台德酸辅助布朗斯台德酸催化下磷酸香豆素对弱亲核试剂的超亲电活化

Zalaltdinova, Alena V; Sadykova, Yulia M; Gazizov, Almir S; Smailov, Atabek K; Syakaev, Victor V; Gerasimova, Daria P; Chugunova, Elena A; Akylbekov, Nurgali I; Zhapparbergenov, Rakhmetulla U; Appazov, Nurbol O; Burilov, Alexander R; Pudovik, Michail A; Alabugin, Igor V; Sinyashin, Oleg G

Cyclic Imines and Their Salts as Universal Precursors in the Synthesis of Nitrogen-Containing Alkaloids

环状亚胺及其盐作为含氮生物碱合成的通用前体

Smolobochkin, Andrey; Gazizov, Almir; Sidlyaruk, Nikita; Akylbekov, Nurgali; Zhapparbergenov, Rakhmetulla; Burilov, Alexander

Discovery of Di(het)arylmethane and Dibenzoxanthene Derivatives as Potential Anticancer Agents

发现二(杂)芳基甲烷和二苯并呫吨衍生物作为潜在的抗癌药物

Smolobochkin, Andrey; Niyazova, Dinara; Gazizov, Almir; Syzdykbayev, Marat; Voloshina, Alexandra; Amerhanova, Syumbelya; Lyubina, Anna; Neganova, Margarita; Aleksandrova, Yulia; Babaeva, Olga; Voronina, Julia; Appazov, Nurbol; Sinyashin, Oleg; Alabugin, Igor; Burilov, Alexander; Pudovik, Michail

Phosphonates of Pectobacterium atrosepticum: Discovery and Role in Plant-Pathogen Interactions.

腐生果胶杆菌的膦酸盐:发现及其在植物-病原体相互作用中的作用

Parfirova Olga, Mikshina Polina, Petrova Olga, Smolobochkin Andrey, Pashagin Alexander, Burilov Alexander, Gorshkov Vladimir

Hybrids of Sterically Hindered Phenols and Diaryl Ureas: Synthesis, Switch from Antioxidant Activity to ROS Generation and Induction of Apoptosis

空间位阻酚类和二芳基脲类化合物的杂合物:合成、从抗氧化活性到活性氧生成及诱导细胞凋亡的转变

Gibadullina, Elmira; Neganova, Margarita; Aleksandrova, Yulia; Nguyen, Hoang Bao Tran; Voloshina, Alexandra; Khrizanforov, Mikhail; Nguyen, Thi Thu; Vinyukova, Ekaterina; Volcho, Konstantin; Tsypyshev, Dmitry; Lyubina, Anna; Amerhanova, Syumbelya; Strelnik, Anna; Voronina, Julia; Islamov, Daut; Zhapparbergenov, Rakhmetulla; Appazov, Nurbol; Chabuka, Beauty; Christopher, Kimberley; Burilov, Alexander; Salakhutdinov, Nariman; Sinyashin, Oleg; Alabugin, Igor

An Unusual Rearrangement of Pyrazole Nitrene and Coarctate Ring-Opening/Recyclization Cascade: Formal CH-Acetoxylation and Azide/Amine Conversion without External Oxidants and Reductants

吡唑氮烯和环状酸酯开环/重环化级联反应的异常重排:无需外部氧化剂和还原剂即可实现形式上的CH-乙酰氧基化和叠氮/胺转化

Chugunova, Elena; Gazizov, Almir S; Islamov, Daut; Matveeva, Victoria; Burilov, Alexander; Akylbekov, Nurgali; Dobrynin, Alexey; Zhapparbergenov, Rakhmetulla; Appazov, Nurbol; Chabuka, Beauty K; Christopher, Kimberley; Tonkoglazova, Daria I; Alabugin, Igor V

Water-Soluble Salts Based on Benzofuroxan Derivatives-Synthesis and Biological Activity

基于苯并呋喃恶烷衍生物的水溶性盐——合成及生物活性

Chugunova, Elena; Matveeva, Victoria; Tulesinova, Alena; Iskanderov, Emil; Akylbekov, Nurgali; Dobrynin, Alexey; Khamatgalimov, Ayrat; Appazov, Nurbol; Boltayeva, Lyazat; Duisembekov, Bakhytzhan; Zhanakov, Mukhtar; Aleksandrova, Yulia; Sashenkova, Tatyana; Klimanova, Elena; Allayarova, Ugulzhan; Balakina, Anastasia; Mishchenko, Denis; Burilov, Alexander; Neganova, Margarita

4,6-Dichloro-5-Nitrobenzofuroxan: Different Polymorphisms and DFT Investigation of Its Reactivity with Nucleophiles

4,6-二氯-5-硝基苯并呋喃恶烷:不同的多晶型及其与亲核试剂反应性的DFT研究

Chugunova, Elena; Akylbekov, Nurgali; Dobrynin, Alexey; Burilov, Alexander; Boga, Carla; Micheletti, Gabriele; Frenna, Vincenzo; Mattioli, Edoardo Jun; Calvaresi, Matteo; Spinelli, Domenico